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2-methanesulfonyl-7-{[2-(methoxymethyl)pyrrolidin-1-yl]sulfonyl}-1,2,3,4-tetrahydroisoquinoline
N-cyclopropyl-5-[3-(1,2-oxazinan-2-yl)propanoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[3-cyclopropyl-1-(3-methylpyridin-4-yl)-1H-1,2,4-triazol-5-yl]-6-(propan-2-yl)pyrimidin-2-amine
N-butyl-5-(4-cyclohexylpiperazine-1-carbonyl)-1-(furan-2-ylmethyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
1'-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-(2-chloro-5-sulfamoylphenyl)-3-{[1-(1H-pyrazol-1-ylmethyl)cyclopropyl]methyl}urea
5-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
2-[(4-phenyl-1,3-thiazol-2-yl)methyl]-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
4-[(diethylamino)methyl]-5-ethyl-N-(4-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)furan-2-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-9-(1-methyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[4-(1,3-benzothiazol-2-yl)piperazine-1-carbonyl]pyridin-3-ol
1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}isoquinoline
(butan-2-yl)({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)(thiophen-3-ylmethyl)amine
1-{1-[1-(propan-2-yl)piperidin-4-yl]piperidin-3-yl}-4-[3-(trifluoromethyl)phenyl]piperazine
5-{2-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-[4-(3-ethyl-1H-indole-2-carbonyl)piperazin-1-yl]pyrazine-2-carbonitrile
8-[(1,3-diphenyl-1H-pyrazol-4-yl)methyl]-1-ethyl-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-amino-6-cyclopropyl-4-(4-hydroxy-3-methylphenyl)pyridine-3-carbonitrile
2-{5-[(2S,4R)-4-hydroxypyrrolidin-2-yl]-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
2-(3-fluoro-4-methoxyphenyl)-2-[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]acetic acid
3-[1-(2H-1,3-benzodioxol-4-ylmethyl)piperidin-3-yl]-N-(4-fluoro-2-methylphenyl)propanamide
1-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-4-(2-methylpyridin-4-yl)-1,4-diazepane
5-({2-[2-(5-chlorothiophen-2-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,4-triazole
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
3-[(2-fluorophenyl)formamido]-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}propanamide
3-chloro-N-(oxan-2-ylmethyl)thiophene-2-carboxamide
3-({[(5-ethylpyridin-2-yl)methyl](methyl)amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
4-[2-amino-3-cyano-6-(1H-pyrrol-2-yl)pyridin-4-yl]benzoic acid
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(5-methyl-1,2-oxazole-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
1-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]cyclopropane-1-carboxamide
4-[(dimethylamino)methyl]-1-[4-(1H-imidazol-1-yl)benzoyl]azepan-4-ol
methyl (2S)-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}pyrrolidine-2-carboxylate
3-[methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amino]propanamide
(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)-N-[3-methyl-1-(2-methylphenyl)-1H-pyrazol-5-yl]pyrrolidine-1-carboxamide
4-{2-[2-(pyridin-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}benzene-1-sulfonamide
2-methyl-1-(1-{[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)propan-1-ol
methyl 3-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-9-(oxan-2-ylmethoxy)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(2-chlorophenyl)-4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-5-methylpiperazin-2-one
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
2-{5-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
2-methoxy-1-(4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1,4-diazepan-1-yl)ethan-1-one
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
methyl[(3-methylquinoxalin-2-yl)methyl][3-(oxolan-2-yl)propyl]amine
5-[(5-{[3-(butan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}furan-2-yl)sulfanyl]-1H-1,2,4-triazole
2-(2-methoxy-6-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}phenoxy)propanoic acid
N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
1-methyl-N-[(5-methyl-1,3,4-thiadiazol-2-yl)methyl]-N-(2-phenylethyl)piperidin-4-amine
3-fluoro-5-methyl-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]imidazo[1,2-a]pyridine-2-carboxamide
N-(2,3-dihydro-1H-inden-1-yl)-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide