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2-(5-fluoro-2-methoxyphenyl)-2-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]acetic acid
N-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)-3-{2-[4-(2-methoxyphenyl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
6-methyl-4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1-[2-(methylsulfanyl)phenyl]piperazin-2-one
4-[(2-chlorophenyl)methyl]-1-(2,5,7-trimethylquinoline-4-carbonyl)-1,4-diazepan-5-one
2-(1H-1,3-benzodiazol-2-ylmethoxy)-1-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
7-(thianthren-1-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
methyl (1R,3S,3aR,6aS)-1-ethyl-5-methyl-4,6-dioxo-3-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-{[(3S,5S)-5-[4-(adamantan-2-yl)piperazine-1-carbonyl]-1-[(2-chloro-6-fluorophenyl)methyl]pyrrolidin-3-yl]sulfanyl}pyrimidine
2-(4-{3-fluoroimidazo[1,2-a]pyridine-2-carbonyl}-1,4-diazepan-1-yl)-1,3-benzothiazole
(1S,5R)-3-[(2-fluoro-5-methoxyphenyl)methyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-[(3-fluorophenyl)methyl]-5-[4-(4-hydroxyphenyl)piperazine-1-carbonyl]piperidin-2-one
4-phenyl-1-[3-(pyridin-4-yl)propanoyl]piperidine-4-carbonitrile
3-methoxy-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylpropanamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]pyrrolidine-3-carboxylic acid
3-propanamido-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)benzamide
methyl 5-{[(2,4-difluorophenyl)methyl]amino}-1-(2-methylpropyl)-3-(pyridine-3-amido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-(3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}phenoxy)ethan-1-ol
1-cyclopropyl-4-[4-(3-methoxyphenyl)piperazine-1-carbonyl]pyrrolidin-2-one
8-methoxy-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-[3-(hydroxymethyl)phenyl]-5-(morpholine-4-sulfonyl)benzoic acid
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-3-(1H-pyrazol-1-yl)benzamide
2-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-1,3-thiazole-4-carboxamide
2-benzyl-9-[(2R)-2-hydroxypropanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-2-(4-fluorophenyl)-1-{4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}ethan-1-one
N-[1-(cyclohexylmethyl)piperidin-3-yl]pyridine-4-carboxamide
4-(morpholin-4-yl)-N-[2-(pyridin-4-yl)ethyl]benzamide
1-[(2,3-dimethoxyphenyl)methyl]-3-hydroxy-3-{[(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
2-(4-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}piperazin-1-yl)acetamide
5-methyl-3-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-3,4-dihydroquinazolin-4-one
2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)-N-cyclopropylacetamide
2-{4-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-4-yl]piperazin-1-yl}phenol
N-[2-(methylsulfamoyl)ethyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
3-fluoro-N-methyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-3-yl}methyl)benzamide
1-[(4-chlorophenyl)methyl]-N-(9H-fluoren-9-yl)-6-oxopiperidine-3-carboxamide
5-fluoro-2-{6-[(2-hydroxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-methyl-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(2-phenylethyl)acetamide
6-ethoxy-4-methyl-2-{4-[(6-methylpyridin-2-yl)methyl]-1,4-diazepan-1-yl}quinazoline
1-ethyl-2-{1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
1-(2-aminoethyl)-N-benzyl-N-(1,3-thiazol-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-2-(pyrrolidin-1-yl)butanamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidine-5-carboxamide
5-{1-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-1H-imidazol-2-yl}-2-methoxyphenol
1-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
2-(3-fluoro-4-hydroxyphenyl)-1-[4-(2-methylphenoxy)piperidin-1-yl]ethan-1-one
1-[(2,3-difluoro-6-methoxyphenyl)methyl]-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
5-{4-[2-(2H-1,3-benzodioxol-5-yl)acetyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
1-[3-(difluoromethoxy)phenyl]-3-[1-(pyrazin-2-yl)piperidin-3-yl]urea
1-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine