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9-[(5-fluoro-2-methoxyphenyl)methyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4-ethylphenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N5-(3-methoxypropyl)-N6-(prop-2-en-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-methoxypropyl)acetamide
(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-4-(thiophene-2-sulfonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(1H-imidazol-4-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-{2-[1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]ethyl}phenol
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-oxo-2,3-dihydro-1H-imidazole-4-carboxamide
1-{2-[4-fluoro-3-(trifluoromethyl)phenyl]pyrimidin-4-yl}piperidin-3-ol
8-[(4-hydroxy-3-methoxyphenyl)methyl]-3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
(1S,5R)-3,6-dibenzyl-3,6-diazabicyclo[3.2.2]nonan-7-one
5-{1-[1-(4-chlorophenyl)cyclopropanecarbonyl]piperidin-4-yl}-5-methyl-3-[2-(morpholin-4-yl)ethyl]imidazolidine-2,4-dione
4-[(1R,7S)-3-(2-ethylbutyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[(2-{1-ethyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)methyl]-1H-pyrazole
5-[3-(benzyloxy)propyl]-2-fluorobenzamide
1-[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)pyrrolidin-3-amine
3-{1-[3-(4-methyl-1,3-thiazol-5-yl)propanoyl]piperidin-4-yl}-N-(3-methylphenyl)propanamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(3-methyl-1H-indol-2-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-6-methylpyridine-3-carboxamide
[(2S,4R)-4-(dimethylamino)-1-[(4-methyl-3,4-dihydro-2H-1,4-benzoxazin-7-yl)sulfonyl]pyrrolidin-2-yl]methanol
(1r,4r)-4-{[(8-fluoroquinolin-2-yl)formamido]methyl}cyclohexane-1-carboxylic acid
1-{2-oxo-2-[2-(pyridin-3-yl)piperidin-1-yl]ethyl}-1,2-dihydropyrimidin-2-one
methyl 6-{[3-(2-phenylpyridin-4-yl)pyrrolidin-1-yl]methyl}pyridine-2-carboxylate
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-5-methylhexanamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}({[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl})amine
2-cyclopropyl-9-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-[(3R,4S)-1-(1H-imidazol-4-ylmethyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
N-[2-(1H-imidazol-4-yl)ethyl]-2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carboxamide
1-[(3-fluorophenyl)methyl]-N-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-6-oxopiperidine-3-carboxamide
2-(4-{[(3R)-3-hydroxypiperidin-1-yl]methyl}phenyl)-6-[2-(1H-pyrazol-1-yl)ethyl]-3,4-dihydropyrimidin-4-one
1-(2-ethyl-2-methyl-4-oxo-3,4-dihydro-2H-1-benzopyran-6-yl)-3-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]urea
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-3-(pyridin-3-yl)propan-1-one
7-(2-methoxyphenyl)-2-(2-phenyl-1,3-oxazol-4-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-({4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
5-[(naphthalen-2-yloxy)methyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
(3S,4R)-1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
(1R,7S)-3-[(3-methoxyphenyl)methyl]-N-methyl-N-(1,2-oxazol-3-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidine-3-carboxamide
dimethyl({[(3S,4R)-4-(propan-2-yl)-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]sulfamoyl})amine
(2S,4R)-4-amino-N,N-diethyl-1-(1,2,3,4-tetrahydroquinoline-8-carbonyl)pyrrolidine-2-carboxamide
methyl 1-{3-[4-({[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]amino}methyl)phenoxy]-2-hydroxypropyl}piperidine-4-carboxylate
4-{6-oxo-1-phenyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1H-pyrazole-3-carboxylic acid
3-fluoro-5-{2-oxo-1-oxa-3,8-diazaspiro[4.6]undecane-8-carbonyl}benzonitrile
4-{1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}pyridine
3,3,3-trifluoro-2-methoxy-N-methyl-2-phenyl-N-(pyrazin-2-ylmethyl)propanamide
N-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)ethyl]piperidine