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(1S,5R)-6-(cyclopropylmethyl)-3-[3-(thiophen-2-yl)propanoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
3-(4-methoxyphenyl)-5-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-1H-pyrazole
6-methoxy-3-({methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]amino}methyl)quinolin-2-ol
2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[1-(thiophen-2-yl)propan-2-yl]acetamide
2-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-4-methylpyrimidine
5-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-2-amine
6-[4-(benzyloxy)piperidine-1-carbonyl]-2-cyclohexyl-1,3-benzoxazole
N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
2-(1-cyclopentyl-3-oxopiperazin-2-yl)-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide
N-(1H-imidazol-2-ylmethyl)-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(2-ethoxyethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
3-[5-(1H-imidazol-2-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-1-(4-methylpiperazin-1-yl)propan-1-one
2-[1-(2,2-dimethylpropyl)-4-[(1-ethyl-1H-indol-3-yl)methyl]piperazin-2-yl]ethan-1-ol
3-(3-fluorobenzoyl)-N-[1-(furan-2-yl)ethyl]-9-methoxy-N-methyl-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[3-(pyridine-3-carbonyl)piperidin-1-yl]propan-1-one
N-{[2-(4-acetylpiperazin-1-yl)-7-methoxyquinolin-3-yl]methyl}-N-(2-methoxyethyl)-1,3-thiazole-5-carboxamide
1-{2-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-ethylpiperidine-4-carboxamide
N-[(1-methyl-1,2,3,6-tetrahydropyridin-4-yl)methyl]-2-(phenylsulfanyl)acetamide
1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-[2-(1H-pyrazol-1-yl)ethyl]piperidine
4-phenyl-1-(1,3-thiazol-4-ylmethyl)azepane
3-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]-1-methyl-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)benzamide
2-(ethylamino)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]pyrimidine-5-carboxamide
N-[1-(furan-2-yl)ethyl]-9-methoxy-7-oxo-3-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
(3aR,6aR)-2-(cyclobutylmethyl)-5-(naphthalene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-({5-[2-(3-fluorophenyl)ethyl]-1,2,4-oxadiazol-3-yl}methyl)-1-methylpiperidine
1-[2-(3-methoxyphenoxy)ethyl]-4-(1-methylpiperidine-4-carbonyl)piperazine
N-[(2-phenyl-1,3-oxazol-4-yl)methyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
N-(2-methyl-2H-1,2,3-triazol-4-yl)-2-(4-methyl-3-phenyl-1H-pyrazol-1-yl)acetamide
5-{1-benzyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-2-methyl-1,3-thiazole
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-3-(1-methyl-1H-pyrazol-4-yl)propanamide
(1S,5R)-3-(1,3-benzoxazol-2-yl)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-(2-{7-[(2-ethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-fluorobenzamide
methyl 2-[(3aR,5R,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-1-methyl-1H-1,3-benzodiazole-5-carboxylate
6-methoxy-N-[2-(1H-pyrrol-1-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-[1-(pent-2-yn-1-yl)piperidin-4-yl]-6-(pyrrolidin-1-yl)pyrimidine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)({[4-methoxy-3-(methoxymethyl)phenyl]methyl})methylamine
3-(2,1,3-benzoxadiazol-5-ylmethyl)-8-methoxy-3,4-dihydroquinazolin-4-one
N-methyl-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)-N-[3-(morpholin-4-yl)propyl]acetamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
N-(cyclohex-1-en-1-ylmethyl)-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-{4-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-1H-1,3-benzodiazole-5-carboxamide
5-methyl-3-{2-oxo-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-[(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)sulfonyl]morpholine-2-carboxylic acid
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-3-{2-[(2-methoxyethyl)(methyl)amino]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-hydroxy-N-(isoquinolin-5-yl)-1,4-oxazepane-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
1-[1-methyl-10-oxo-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecane-4-carbonyl]cyclopropane-1-carboxamide
5-[2-(aminomethyl)piperidine-1-carbonyl]-2-(3,5-dichlorophenyl)pyrimidin-4-ol