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1-[2-chloro-5-(morpholine-4-carbonyl)phenyl]-3-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]urea
N-(3-{[(2-methylpropyl)(pyridin-2-ylmethyl)carbamoyl]methoxy}phenyl)propanamide
N-(1H-1,3-benzodiazol-2-yl)-2-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]acetamide
2-[3-(3-fluoro-4-methoxyphenyl)-1H-indazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
7-(1-benzothiophen-3-yl)-4-(4-methyl-1H-imidazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-1-(3,4-dihydro-2H-1-benzopyran-2-carbonyl)piperidine
2-(oxolan-2-ylmethyl)-8-(quinoline-6-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
3-{[4-(pyridin-2-ylmethyl)-1,4-diazepan-1-yl]methyl}benzoic acid
8-cyclopropanecarbonyl-2-[2-(4-fluorophenyl)acetyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[1-(1,4-dithiepan-6-yl)piperidin-3-yl]methyl}-4-phenylbenzamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-2-(dimethyl-1,3-thiazol-5-yl)acetamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1,4-diazepane
2-(adamantan-1-yl)-4-hydroxy-N-(1-methyl-6-oxopiperidin-3-yl)pyrimidine-5-carboxamide
N,N,5,7-tetramethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
1-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
(cyclohex-3-en-1-ylmethyl)(2-methoxyethyl)({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)amine
3-ethyl-1-methyl-4-({3-methyl-1-[2-(4-methylpiperazin-1-yl)ethyl]-1H-pyrazol-4-yl}methyl)piperazin-2-one
3-(1H-1,2,3-benzotriazol-1-yl)-N-[2-(1-methylpiperidin-3-yl)ethyl]propanamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
9-(3-chloro-4-fluorobenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-2-(morpholin-4-yl)-2-oxoacetamide
N-ethyl-2-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}pyrimidin-4-amine
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl){[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
(3ar,6ar)-N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-{3-[(1-cyclopentanecarbonylpiperidin-4-yl)oxy]benzoyl}morpholine
5-(oxolan-2-yl)-N-{2-[(pyridin-3-yl)amino]ethyl}thiophene-2-carboxamide
1-{5-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1H-pyrazole-3-carbonyl}-4-(cyclopropylmethyl)piperazine
3-[({[3-(cyclopentyloxy)phenyl]methyl}amino)methyl]-N,N-dimethylpyridin-2-amine
2-(methylamino)-N-{[1-(2-methylphenyl)pyrrolidin-3-yl]methyl}acetamide
N-[(2R,3R)-1'-(2,4-difluorobenzoyl)-2-(pyridin-2-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-methylacetamide
2-fluoro-N-methyl-5-({[(4-methyl-1,4-oxazepan-6-yl)methyl]carbamoyl}amino)benzamide
N-(pyridin-4-ylmethyl)-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
N-[(3R,4S)-1-(oxan-4-yl)-4-propylpyrrolidin-3-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butanamide
4-(1,4-oxazepane-4-carbonyl)-1,2-dihydroquinolin-2-one
N3-benzyl-1-cyclopropyl-N5-[(2,4-difluorophenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-1,5-dimethyl-1H-indole-2-carboxamide
1-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-2-[5-(oxolan-2-yl)thiophen-2-yl]-1H-imidazole
N-[2-(dimethylamino)ethyl]-3-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-4-yl)propanamide
methyl 4-(5-{[3-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-3-(1,2-oxazolidin-2-yl)propanamide
2-ethyl-5-{[4-(2-phenoxyethyl)piperazin-1-yl]methyl}pyrimidine
5-{1-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-1H-1,2,3-triazol-4-yl}-N,N-dimethylpyrimidin-2-amine
1-(4-{[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
1-{5-[(3-methyl-1-benzofuran-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carbonyl}pyrrolidine
3-methanesulfonamido-N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)propanamide
N-[2-(trifluoromethyl)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
2-amino-3-ethyl-N-[2-(2-methylphenyl)ethyl]-3H-imidazo[4,5-b]pyridine-6-carboxamide
(2R,3R,6R)-3-(4-methylphenyl)-5-(4-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane