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(4aR,8aS)-6-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1-[3-(2-oxopyrrolidin-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
8-[2-chloro-5-(trifluoromethyl)benzoyl]-2,8-diazaspiro[4.5]decan-3-one
1-ethyl-7-methyl-3-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]-1,4-dihydro-1,8-naphthyridin-4-one
2-[5-({4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]pyrazine
2-methoxy-N-[7-methoxy-4-(2-methoxypyridin-3-yl)-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]acetamide
1-[1-(1-cyclopropanecarbonylpiperidin-4-yl)piperidine-3-carbonyl]-1,2,3,6-tetrahydropyridine
({1-[(2-fluorophenyl)methyl]-2-methanesulfonyl-1H-imidazol-5-yl}methyl)(methyl)(2-phenylethyl)amine
3-(1-cyclohexyl-1H-pyrazol-5-yl)-1-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
4-[7-(oxolane-2-amido)-1,2,3,4-tetrahydroisoquinoline-2-carbonyl]pyridin-1-ium-1-olate
1'-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({8-[(4-fluoro-3-methoxyphenyl)methyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)-2-methyl-1,3-thiazole-4-carboxamide
2-amino-6-cyclopropyl-4-[3-(1H-pyrazol-1-yl)phenyl]pyridine-3-carbonitrile
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-3-yl)propanamide
2-{2-[1-(propan-2-yl)piperidin-4-yl]acetamido}-2-[2-(trifluoromethyl)phenyl]acetic acid
3-(2-methylpiperidin-1-yl)-N-[4-(1H-pyrazol-5-yl)phenyl]azetidine-1-carboxamide
8-(furan-2-ylmethyl)-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,5-dimethylphenyl)methyl]-4-methyl-1,4-diazepan-5-one
2-{1-[(3-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(1H-pyrazol-4-yl)ethyl]acetamide
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)acetamide
4-cyclobutyl-6-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]pyrimidin-2-amine
3-{[(1-methyl-1H-imidazol-2-yl)methyl]sulfamoyl}-N-[(2S)-pyrrolidin-2-ylmethyl]benzamide
N4-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-2-methylpyrimidine-4,6-diamine
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methylpropanamide
1-{2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methyl-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
5-(6-{[2-(dimethylamino)ethyl]amino}-1H-pyrrolo[2,3-b]pyridin-4-yl)-1,3-benzothiazol-2-amine
(5R)-5-({5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)pyrrolidin-2-one
4-[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)amino]-5-methyl-N-[3-(morpholin-4-yl)propyl]thieno[2,3-d]pyrimidine-6-carboxamide
2,4-difluoro-3-methoxy-N-{2-[(3-methylpyridin-4-yl)amino]ethyl}benzamide
methyl 6-[(3aS,6aR)-3-[2-(4-methoxyphenyl)ethyl]-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-5-yl]pyridine-3-carboxylate
1-(2H-1,3-benzodioxol-5-yl)-5-[2-(1H-imidazol-1-yl)ethyl]-3-(2-phenylethyl)-1H-1,2,4-triazole
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carboxamide
methyl 1-({1-[(2,3-difluorophenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)piperidine-4-carboxylate
2-(4-fluorophenyl)-4-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}morpholine
N-{1-[7-(1-benzothiophen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}furan-2-carboxamide
4-hydroxy-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-(3-methylphenyl)pyrimidine-5-carboxamide
ethyl 4-{[4-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
methyl 1-benzyl-3-cyclopropaneamido-5-{[(2-methoxyphenyl)methyl]amino}-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(1-methoxypropan-2-yl)amine
1-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
4-{4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}morpholine
5-acetyl-N-benzyl-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-amino-7-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-6-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
1-[1-(2-hydroxyethyl)piperidine-3-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-(2-aminoethyl)-5,6-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
2-(3-chloro-6-oxo-1,6-dihydropyridazin-1-yl)-N-[2-(2-ethylphenoxy)ethyl]-N-methylacetamide
7-(2-hydroxyethyl)-2-[5-(trifluoromethyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
2-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}thiophen-3-amine