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N-[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]-2-methoxypyridine-4-carboxamide
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
5-(2-chloro-4-methoxyphenoxymethyl)-N-[1-(propan-2-yl)cyclopropyl]-1H-pyrazole-3-carboxamide
(3aS,7aR)-2-(2-methoxy-6-methylbenzoyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]pyrimidin-2-amine
3-[(3R,4R)-3-(hydroxymethyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidine-1-carbonyl]benzonitrile
4-benzyl-3-ethyl-1-(morpholine-4-sulfonyl)-1,4-diazepan-5-one
4-(furan-2-yl)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
5-[(1-tert-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
(3S,5R)-5-[(pyridin-4-ylmethyl)carbamoyl]-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine-3-carboxylic acid
N-({7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)pyridine-2-carboxamide
4-(1-benzylpyrrolidin-3-yl)-4H-1,2,4-triazole
2-[({1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}oxy)methyl]pyridine
1-{[5-(hydroxymethyl)furan-2-yl]methyl}-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
3-[({[(2S)-5-oxopyrrolidin-2-yl]methyl}(pyridin-2-ylmethyl)amino)methyl]-1,2-dihydroquinolin-2-one
3-[(5-phenyl-1,2,4-oxadiazol-3-yl)methyl]-1,3-diazinane-2,4-dione
N-[1-(carbamoylmethyl)piperidin-4-yl]-4-[(diethylamino)methyl]-5-ethylfuran-2-carboxamide
1-{[2-(dimethylamino)-1,3-thiazol-5-yl]methyl}-N-[4-(furan-2-yl)phenyl]piperidine-3-carboxamide
(2R,3R,6R)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane
N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}thian-4-amine
6-amino-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]pyridine-3-carboxamide
N,1-dimethyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}azepane-2-carboxamide
1-[2-(dimethylamino)ethyl]-4-ethyl-3-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-[4-(morpholin-4-ylmethyl)phenyl]urea
2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-4-(1H-pyrazol-1-ylmethyl)-1,3-oxazole
(3aR,5R,6S,7aS)-2-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-octahydro-1H-isoindole-5,6-diol
2-(2H-1,3-benzodioxole-5-carbonyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
(2S)-1-[(5-cyano-1H-pyrrol-3-yl)methyl]-N-[4-(3-methoxyphenyl)phenyl]pyrrolidine-2-carboxamide
N-cyclopropyl-2,4-difluoro-3-methoxy-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
N-(2-methylpropyl)-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
N-methyl-N-[(5-methylfuran-2-yl)methyl]-2,3,4,9-tetrahydro-1H-carbazole-1-carboxamide
(4aS,8aR)-1-butyl-6-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
5-(3-fluoropyridin-4-yl)-8-methoxyquinoline
2-[3-(hydroxymethyl)-3-(3-methylbut-2-en-1-yl)piperidine-1-carbonyl]benzonitrile
4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-methanesulfonylpiperidine
N-{2-[({5-[(dimethylamino)methyl]furan-2-yl}methyl)sulfanyl]ethyl}-1-methyl-1H-indole-6-carboxamide
3-[(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-2,2-dimethylpropan-1-ol
6,8-dimethyl-4-(pyridin-4-yl)quinoline
3-[2-(piperazin-1-ylmethyl)phenyl]quinoline
3-(1,4-dioxan-2-ylformamido)-N-(3-methylphenyl)propanamide
1-(4-aminopyrimidin-2-yl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylic acid
2-[3-(5-methylfuran-2-yl)-5-[(2-oxopyrrolidin-1-yl)methyl]-1H-1,2,4-triazol-1-yl]benzoic acid
3-[(pyridin-2-ylmethyl)sulfamoyl]-5-(pyrimidin-5-yl)benzoic acid
1-[4-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)piperidin-1-yl]ethan-1-one
1-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-(pyrrolidin-1-yl)ethane-1,2-dione
[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl]methanol
3-(3-ethoxypropanamido)-4-(3-methylpiperidin-1-yl)benzamide
1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]ethan-1-one
3-methoxy-6-{4-[1-(piperidin-1-yl)ethyl]phenyl}pyridazine