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2-(pyridin-2-ylmethyl)-8-(pyridine-2-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
2-[3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyridine-3-carboxylic acid
4-{2-[3-(4-chlorophenyl)piperidin-1-yl]-2-oxoethyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1-[3-({[3-(propan-2-yloxy)propyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
2,4-dimethyl-5-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1H-pyrrole-3-carboxylic acid
2-[(3S)-3-hydroxypyrrolidin-1-yl]-1-methyl-N-[2-(pyridin-4-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
N-[3-(benzylsulfanyl)propyl]-3-(1H-imidazol-2-yl)benzamide
N,2-dimethyl-N-(quinolin-5-ylmethyl)-1,3-benzothiazole-5-carboxamide
1'-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}acetamide
{[2-(furan-2-yl)phenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-(4-chloro-1-methyl-1H-pyrrole-2-carbonyl)-7-propyl-2,7-diazaspiro[4.5]decan-6-one
4-[(2-chlorophenyl)methyl]-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
3-[(3R,4S)-4-(dimethylamino)-1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-3-yl]propan-1-ol
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[4-(2-methylpropyl)benzoyl]-decahydro-1,6-naphthyridin-2-one
2-{4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridine-3-carboxamide
N,N-dimethyl-5-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-3-carboxamide
4'-[(3,5-dimethoxyphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[4-(2-acetamidoacetamido)-2-methylphenyl]-2,2-dimethylpropanamide
N-(2-methoxyethyl)-1-[1-(6-methylpyridazin-3-yl)piperidin-4-yl]piperidine-3-carboxamide
N-(2-hydroxyethyl)-N-methyl-2-[methyl(2-phenylethyl)amino]-2,3-dihydro-1H-indene-2-carboxamide
11-{[(2,3-difluorophenyl)methyl]amino}-4-(2,3-dihydro-1H-inden-2-yl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[4-(methylsulfanyl)phenyl]methyl})amine
2-(2,5-dioxoimidazolidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)acetamide
N,1-dimethyl-N-{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-{1-[6-amino-2-(diethylamino)pyrimidin-4-yl]piperidin-4-yl}methanesulfonamide
1-benzyl-N-(cyclopropylmethyl)-2-methyl-5-(2-methylpropanamido)-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-7-carboxamide
1-(2,3-dimethyl-1H-indole-5-carbonyl)-N-(4-methoxyphenyl)piperidin-3-amine
4-[(1S,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-1-phenylbutan-1-one
2-({3-[4-(2,4-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-3-methoxyphenol
N-(1-{1-[(2,5-dimethoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2,2-dimethylpropanamide
[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
2,5-dimethyl-N-[3-(1H-1,2,4-triazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-1-(2-benzylmorpholin-4-yl)ethan-1-one
1-(2,3-dimethylphenyl)-4-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazine
4-methyl-5-[3-(2-methylphenoxy)azetidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-6-methylpyridine-3-carboxamide
1-[2-methyl-5-(thiomorpholine-4-carbonyl)phenyl]imidazolidin-2-one
3-(2-phenylethyl)-5-[1-(prop-2-en-1-ylsulfanyl)ethyl]-1H-1,2,4-triazole
5-acetyl-N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methylthiophene-3-carboxamide
4-(naphthalen-2-yloxy)-1-(oxolan-3-ylmethyl)piperidine-4-carboxylic acid
5-ethyl-2-{1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-imidazol-2-yl}pyridine
4-(naphthalen-2-yloxy)-1-[(1-propyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxylic acid
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[1-(pyrimidin-4-yl)ethyl]acetamide
4-(2-methylphenoxy)-1-(thiophene-2-carbonyl)piperidine-4-carboxylic acid
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-methylpyrimidine
[2-({4-[(2,3-difluoro-6-methoxyphenyl)methyl]piperazin-1-yl}methyl)phenyl]methanol
5-({3-[3-(2-methylphenyl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)isoquinoline
4-cyano-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
4-{5-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}phenol