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3-(1-benzothiophen-3-yl)pyridin-2-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
methyl({[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})[2-(pyridin-2-yl)ethyl]amine
6-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-(morpholin-4-yl)pyrimidin-4-amine
(1-{[2-(3-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)(thiophen-2-yl)methanol
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl](methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
5-acetyl-N-(2-hydroxy-2-phenylethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
1-(3-chlorophenyl)-4-[1-(thian-4-yl)piperidin-3-yl]piperazine
4-(1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-4-carbonyl)morpholine
3-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
(5S,9aS,9bS)-5-[3-(2-methylphenyl)phenyl]-2-(1-methylpiperidin-4-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
methyl (2S,4R)-1-[(4-methoxy-2,5-dimethylphenyl)methyl]-4-(2-methylpropanamido)pyrrolidine-2-carboxylate
1-(2-methyl-1,3-thiazole-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-[1-(methoxymethyl)cyclobutanecarbonyl]-4-(pyridin-4-yl)piperazine
3-(4-{[4-(oxan-4-yl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({imidazo[1,2-a]pyrimidin-2-ylmethyl})amine
4-(4-methyl-1H-pyrrole-2-carbonyl)-1-[(4-methylphenyl)methyl]piperazin-2-one
6-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidine-1-carbonyl]-1,3-dimethyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{[4-(dimethylamino)oxan-4-yl]methyl}-3-(isoquinolin-5-yl)urea
N-[3-(pyridin-3-yl)propyl]-1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
7-cyclohexyl-2-[(3,4-dimethoxypyridin-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
[2-(2-chlorophenyl)ethyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[2-(4-{[2-(1H-indol-3-yl)acetamido]methyl}-5-methyl-1,3-oxazol-2-yl)phenyl]pyridine-2-carboxamide
1-[(2S)-oxolane-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{[1-(dimethylsulfamoyl)-4-hydroxyazepan-4-yl]methyl}-2,5-dimethylfuran-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
2-(1,2-oxazol-5-yl)-4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
4-(1H-pyrazol-1-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
(1R,9aR)-1-(2-methoxy-4-methylphenoxymethyl)-octahydro-1H-quinolizine
4-(3-methoxypyrazin-2-yl)piperazin-2-one
8-(6-methoxypyrimidin-4-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-1-(4-methoxyphenyl)piperazin-2-one
N-(2,6-dimethylphenyl)-3-[3-(pyridin-3-yl)propanamido]benzamide
{[2-(4-fluoro-3-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)propylamine
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-phenyl-1,2-oxazole-4-carboxamide
1-{1-[4-methyl-6-(methylsulfanyl)quinolin-2-yl]piperidin-4-yl}piperidin-4-ol
(4aS,7aR)-1-(3-methylbenzoyl)-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(3-{2-hydroxy-3-[methyl(propan-2-yl)amino]propoxy}-4-methoxyphenyl)methyl]-1λ6-thiomorpholine-1,1-dione
propyl (2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxylate
1-(3,4-difluorobenzoyl)-N-(3,4-dimethylphenyl)piperidin-3-amine
2-(2-methyl-1,3-thiazol-4-yl)-1-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethan-1-one
3-(4-methylthiophen-2-yl)-N-[3-(morpholin-4-yl)propyl]-5-(morpholine-4-sulfonyl)benzamide
2-[4-(2-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-[1-(pentan-3-yl)-1H-pyrazol-5-yl]acetamide
2-{4-[(2S,4R)-4-aminopyrrolidine-2-carbonyl]piperazin-1-yl}-1-(piperidin-1-yl)ethan-1-one
1-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}-4-methyl-1H-pyrazole
N,N-diethyl-1-({4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl}methyl)piperidine-3-carboxamide
3-cyclobutyl-5-[(8-methoxy-2H-chromen-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
1-{[(3R,4R)-1-[6-amino-2-(methylsulfanyl)pyrimidin-4-yl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
2-{2-[1-(5-aminopentyl)-4-phenyl-1H-imidazol-5-yl]phenoxy}ethan-1-ol