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N-(3-oxo-3-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propyl)methanesulfonamide
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]piperidine
(2R)-N-{2-[(2-ethylphenyl)carbamoyl]phenyl}-5-oxopyrrolidine-2-carboxamide
methyl 3-(2-methoxybenzamido)-5-[(pyrazin-2-ylformamido)methyl]benzoate
N-[2-(4-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]-1-(oxan-4-yl)piperidine-3-carboxamide
1-methyl-N-({5-[4-(methylsulfanyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-5-carboxamide
N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-(pyridin-3-yl)pyrimidin-2-amine
(5S,9aS,9bS)-5-[(E)-2-(furan-2-yl)ethenyl]-2-(3-methoxyphenyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-(1-{7-[(9-ethyl-9H-carbazol-3-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-3-methoxypropanamide
6-(2-methoxy-2-phenylacetyl)-N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4,6-dimethyl-5-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]pyrimidin-2-amine
1-[3-(2-ethylphenoxy)azetidin-1-yl]-2-(1-ethylpiperidin-4-yl)ethan-1-one
4-fluoro-3-hydroxy-N-(pyrimidin-4-ylmethyl)benzamide
{5-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decane-4-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
[(3R,4S)-1-[(2,3-difluorophenyl)methyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[3-(methylsulfanyl)phenyl]methyl}acetamide
2-[1-methyl-4-(quinolin-5-ylmethyl)piperazin-2-yl]ethan-1-ol
1-({5-[1-(thiophen-2-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]thiophen-3-yl}methyl)pyrrolidine
N-[(5-methylpyrazin-2-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
5-{1-[(2,4-dimethylphenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
1-[2-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-oxoethyl]azepan-2-one
N-[(5-methylfuran-2-yl)methyl]-3-(pyridin-4-yl)propanamide
N-ethyl-N-[2-(morpholin-4-yl)ethyl]-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(4aR,7aS)-1-{2-[4-(2-hydroxyethyl)piperidin-1-yl]pyrimidin-4-yl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cyclopentyl-N-{2-[ethyl(3-methylphenyl)amino]ethyl}-6-oxopiperidine-3-carboxamide
(1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)methanol
3-(2-ethyl-1H-imidazol-1-yl)-1-[(2S,6S)-6-(hydroxymethyl)-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]propan-1-one
N-[(dimethyl-1,3-thiazol-5-yl)methyl]-1-(2-ethoxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-[2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carbonyl]azepane
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
9-(1,4-dithiepan-6-yl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1'-(2-hydroxypyridine-3-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(2-{[4-(dimethylamino)-5-methylpyrimidin-2-yl]amino}ethyl)pyridine-3-carboxamide
N-[cyclopropyl(pyridin-2-yl)methyl]-1-[(2,6-difluorophenyl)methyl]-N-methyl-1H-1,2,3-triazole-4-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-[(1S,4S)-3,3-dimethyl-2-methylidenebicyclo[2.2.1]heptane-1-carbonyl]piperidine
N-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-2-(pyridin-2-yl)pyrrolidine-1-carboxamide
{1-[1-(4-fluorophenyl)piperidin-4-yl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
4-cyclobutanecarbonyl-2-(2,2-diphenylethyl)morpholine
(3R,4R)-4-cyclobutyl-3-methyl-1-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidin-4-ol
1'-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
8-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-methyl-1-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(4-methylphenyl)-1,2-oxazol-3-yl]methyl}-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
N-ethyl-3,6-dimethyl-N-(propan-2-yl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
1-[2-({[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}amino)-4-methylpyrimidin-5-yl]ethan-1-one
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
3-[(dimethylamino)methyl]-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)benzamide
1-cycloheptyl-N-[1-(pyridin-4-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
(4-methyl-5-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}-4H-1,2,4-triazol-3-yl)methanol