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1-(1,2,3,4-tetrahydroisoquinolin-2-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butan-1-one
4-[2-(2-{[4-(pyrrolidin-3-yl)piperazin-1-yl]methyl}phenoxy)ethyl]morpholine
2-(2-phenylethyl)-1-{[2-(pyrrolidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperidine
3-methyl-6-{5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-1,2,4-oxadiazol-3-yl}pyridazine
2-{[(1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)oxy]methyl}pyridine
(2S,3R)-2-({[2-chloro-5-ethoxy-4-(propan-2-yloxy)phenyl]methyl}amino)-3-hydroxybutanamide
4-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
3-(2-{7-[ethoxy(phenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}-2-oxoethyl)-1,3-oxazolidin-2-one
N3-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidine-1,3-dicarboxamide
4-(2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}morpholine-4-carbonyl)-2,6-dimethylquinoline
(4aS,7aR)-1-(4-methyl-2-oxopentanoyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-methyl-2-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]pyrrolidin-2-yl}-1H-1,3-benzodiazole
2-({2,3-dimethyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)acetamide
3-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}pyridine
1-{4-[(2-fluorophenyl)methyl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
2-{3-[(2-methoxyphenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazol-1-yl}pyridine
N-(2,4-dimethylphenyl)-3-[4-(methylsulfanyl)benzoyl]piperidine-1-carboxamide
N-(cyclopropylmethyl)-2-(2-hydroxyacetyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
9-methoxy-7-(6-methoxypyridin-2-yl)-4-(1H-pyrrol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(1S,5R)-3-(1-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-butyl-4-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]-1-methylpiperazin-2-one
7-(2,3,4-trimethoxyphenyl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine
4-{2-cyclobutyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[5-(methoxymethyl)furan-2-carbonyl]piperidine
2-[4-({4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[3-(piperidin-1-yl)propyl]amine
1-(cyclopropylmethyl)-3-hydroxy-3-({[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]amino}methyl)piperidin-2-one
N-(butan-2-yl)-N-cyclopentyl-2-methanesulfonylacetamide
N-[2-(benzylsulfanyl)ethyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]amine
N-[(3-methoxyphenyl)methyl]-N-methyl-2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]acetamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}pyrazolo[1,5-a]pyridine-7-carboxamide
(3aS,6aS)-2-(ethanesulfonyl)-5-{[4-(methylsulfanyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]cyclopentanecarboxamide
1-cyclopentanecarbonyl-N-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-4-amine
8-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
8-(5-phenoxyfuran-2-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-[(3,4-dimethoxyphenyl)methyl]-N-(oxan-4-yl)-1,3-benzoxazole-6-carboxamide
(1R,3S)-3-{cyclopentyl[(2,4-dimethoxyphenyl)methyl]carbamoyl}cyclopentane-1-carboxylic acid
N-[2-(1H-imidazol-1-yl)-1-phenylethyl]-1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(4-methoxyphenyl)-3-[1-(propan-2-yloxy)ethyl]-4H-1,2,4-triazole
6-{[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]methyl}-2-oxo-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1,2-dihydropyridine-3-carboxamide
(2E)-3-(pyridin-4-yl)-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}prop-2-en-1-one
(3aS,6aS)-2-(cyclopropylmethyl)-5-{[2-(methylsulfanyl)phenyl]methyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-methyl-1,3-oxazole-4-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(pyridin-3-yl)piperazine
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[4-(propan-2-yl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
1-[(2,4-dimethoxyphenyl)methyl]-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
methyl 1-[(3R,5S)-5-{[2-(4-fluorophenyl)ethyl]carbamoyl}-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N-methyl-N-{[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl}cyclohexanamine
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-1-[6-methyl-2-(piperidin-1-yl)pyrimidin-4-yl]piperidin-4-amine