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1-[2-(4-phenylpiperidin-1-yl)acetyl]piperidine-3-carbonitrile
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetamide
4-{3-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]phenyl}-4H-1,2,4-triazole
N-butyl-2-methanesulfonamido-N-[(3-methoxyphenyl)methyl]propanamide
9-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(2-ethyl-7-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
1-(3-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-3-methylbut-2-en-1-one
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(3-fluorophenyl)methyl]-N-[(2-methoxyphenyl)methyl]pyrrolidine-2-carboxamide
(2S)-N-ethyl-1-(6-ethyl-2-oxo-1,2-dihydropyridine-4-carbonyl)pyrrolidine-2-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(2-chlorophenoxy)piperidin-1-yl]ethan-1-one
N-[4-(2,6-dimethylphenyl)phenyl]-2-methoxyacetamide
ethyl 5-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-methoxy-4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
N-[1-(pyrimidin-4-yl)ethyl]thieno[2,3-d]pyrimidin-4-amine
1-(5,6,7,8-tetrahydronaphthalen-1-yl)-3-[2-(1,3-thiazol-4-yl)ethyl]urea
4-[4-chloro-2-(1,2-oxazolidine-2-carbonyl)phenoxy]-1-cyclopentylpiperidine
N-(furan-2-ylmethyl)-N-(1-hydroxybutan-2-yl)-1-methyl-1H-pyrrole-2-carboxamide
2-methyl-N-{[4-(3-oxo-4-phenylpiperazine-1-carbonyl)phenyl]methyl}propanamide
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
2-amino-8-{8-oxatricyclo[7.4.0.02,7]trideca-1(9),2(7),3,5,10,12-hexaen-6-yl}-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-{2-ethyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-2-methoxyethan-1-one
4-{5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]-1H-pyrazol-3-yl}phenol
2,6-dimethyl-3-[3-(propoxymethyl)pyrrolidine-1-carbonyl]quinoline
6-methyl-N-[1-(thian-4-yl)piperidin-4-yl]imidazo[2,1-b][1,3]thiazole-5-carboxamide
N-{[4-(aminomethyl)phenyl]methyl}-2-(1-methylpyrrolidin-2-yl)acetamide
4-chloro-2-methoxy-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}benzamide
N-cyclobutyl-5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-1,3-benzoxazole-5-carboxamide
(3S,4R)-4-methyl-1-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidine-4-carbonyl}piperidine-3,4-diol
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-(1-cycloheptylpiperidin-3-yl)-3,4-dimethoxybenzamide
(3R)-1-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]pyrrolidin-3-ol
4-{6-[2-(3,5-dimethyl-1H-pyrazol-1-yl)-4-methylphenyl]pyrazine-2-carbonyl}morpholine
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-N5-(oxolan-2-ylmethyl)-1-(2-phenylethyl)piperidine-3,5-dicarboxamide
3-{[(cyclopropylmethyl)(propan-2-yl)amino]methyl}benzonitrile
8-(6-fluoro-2-oxo-1,2-dihydroquinoline-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(3S,5S)-5-[(6-methylpyridin-3-yl)carbamoyl]-1-(oxan-4-yl)piperidine-3-carboxylic acid
4-[1-(2-phenylbenzoyl)azetidin-3-yl]pyridine
N-{[5-(6-methoxypyridazin-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyrimidin-2-ylsulfanyl)acetamide
N-methyl-1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-(thiophen-3-ylmethyl)piperidine-4-carboxamide
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
2-(1H-imidazol-1-yl)-1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
N-[3-(hydroxymethyl)phenyl]-5-{1-[(2E)-4-methylpent-2-en-1-yl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[(4-methylphenyl)(pyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
{3-[(2-fluorophenyl)methyl]-1-(2-phenylethyl)piperidin-3-yl}methanol
N-({7-[(2-chloro-4,5-dimethoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-2,5-dimethylfuran-3-carboxamide
(3R)-1-[6-(thiomorpholin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]pyrrolidin-3-ol
N-methyl-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(oxan-4-yl)ethyl]acetamide
7-cyclohexyl-2-(pyridin-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one