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4-(2-ethoxyphenyl)-3-[(methylamino)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
(3R,4S)-4-cyclopropyl-1-{[5-(dimethyl-1,2-oxazol-5-yl)furan-2-yl]sulfonyl}pyrrolidin-3-amine
5-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane-1-carbonyl]quinoline
5-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
4-[3-(4H-1,2,4-triazol-4-yl)phenyl]phenol
3-(pentan-2-yl)-8-[2-(piperidin-1-yl)acetyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-1-(cyclohexylmethyl)-N-methyl-6-oxopiperidine-3-carboxamide
2-{3-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]phenoxy}acetamide
1-(4,7-dimethylquinazolin-2-yl)-N-(2-methylpropyl)piperidine-4-carboxamide
4-{2-methyl-1-[4-(4H-1,2,4-triazol-3-yl)piperidin-1-yl]propan-2-yl}morpholine
N-[2-(4-hydroxyphenyl)-2-oxoethyl]-N-methyl-3-(morpholin-4-yl)benzamide
1-[(2S)-2-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrrolidin-1-yl]ethan-1-one
1-[(4-chlorophenyl)methyl]-4-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}piperazine
N-[1-(3-methoxyphenyl)ethyl]-N-methylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-(1-{4-[(1S,5R)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl]phenyl}-1H-pyrazol-4-yl)pyridine-3-carboxamide
2-ethoxy-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}acetamide
3-(1H-1,3-benzodiazol-2-yl)-1-[3-hydroxy-3-(2-methylphenyl)pyrrolidin-1-yl]propan-1-one
2-(5-acetylthiophen-3-yl)-N-[(1-benzylpiperidin-4-yl)methyl]-N-methylacetamide
3-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-N-(pyridin-3-ylmethyl)propanamide
7-methoxy-3-[(4-methyl-1,4-diazepan-1-yl)methyl]-2-(thiophen-2-yl)quinoline
1-(1H-1,2,4-triazole-3-carbonyl)-4-[(2,4,6-trimethoxyphenyl)methyl]piperazine
N-[(1-{[1-(2-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]thiophene-2-carboxamide
3-{1-[2-(adamantan-1-yl)acetyl]piperidin-4-yl}-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-1-benzyl-4-[(2,3-dihydro-1H-inden-2-yl)amino]-N-[2-(2-fluorophenyl)ethyl]pyrrolidine-2-carboxamide
N-methyl-N-(1-{[5-methyl-2-(3-phenoxyphenyl)-1,3-oxazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(propan-2-yl)acetamide
1-methyl-3-propyl-N-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-1H-pyrazole-5-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({[(2-methyl-1H-indol-5-yl)methyl]amino}methyl)piperidin-2-one
2-amino-6-tert-butyl-4-[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]pyridine-3-carbonitrile
6-methoxy-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,3-benzothiazol-2-amine
3-[1-(1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]benzoic acid
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(hydroxymethyl)azepan-4-ol
1-{2-[(2,6-dichlorophenyl)methyl]-4-hydroxypyrimidine-5-carbonyl}piperidine-4-carboxylic acid
N-(1-{1-[(4-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
7-fluoro-3-({methyl[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]amino}methyl)-1-(pyridin-3-ylmethyl)-1,2-dihydroquinolin-2-one
2-(2,3-dihydro-1H-inden-1-yl)-N-[3-(pyridin-4-yl)propyl]acetamide
1-(2-methylpropyl)-4-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidine
[3-(methylsulfanyl)butyl][(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
1-(azepan-1-yl)-3-[3-({[(5-fluoro-2-methylphenyl)methyl]amino}methyl)phenoxy]propan-2-ol
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-(2-chloro-5-methylphenyl)-3-[3-(methylsulfanyl)propyl]urea
4-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}benzoic acid
(2S,4R)-1-(adamantan-2-yl)-N-{imidazo[1,2-a]pyridin-2-ylmethyl}-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
(4aR,7aS)-1-butanoyl-4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-4-methylpentane-1,2-dione
N-(butan-2-yl)-1-methyl-N-(pyridin-4-ylmethyl)-1H-indazole-3-carboxamide
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl})amine
dimethyl[2-(4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}morpholin-2-yl)ethyl]amine