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2-{1-[(2-ethoxyphenyl)methyl]-4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-2-yl}ethan-1-ol
4-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
(1-cyclopropylethyl)({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-[1-(4-methoxyphenyl)ethyl]-N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
ethyl 2-{1-[2-(1H-1,2,4-triazol-1-yl)acetyl]piperidin-2-yl}acetate
1-cyclopentyl-3-(3-fluorophenyl)-3-{2-[(2S)-4-methyl-2-(propan-2-yl)piperazin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
N-[2-(4-chlorophenyl)ethyl]-2-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-4-(3-hydroxy-3-methylbutyl)benzamide
2-benzyl-8-(1,3-thiazol-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[1-(1H-indole-6-carbonyl)piperidin-3-yl]-4-methyl-1H-1,3-benzodiazole
6-{[(3R,4S)-1-(cyclopropanesulfonyl)-4-(propan-2-yl)pyrrolidin-3-yl]amino}pyridine-2-carbonitrile
2-{methyl[7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
3-{2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamido}propanamide
(1S,5R)-6-(2-methoxyethyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{1-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}piperidin-3-ol
7-{[4-(pyridin-2-yl)piperazin-1-yl]methyl}-4-(thian-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-(4-{[(3S)-3-(dimethylamino)azepan-1-yl]methyl}phenoxy)-1-(morpholin-4-yl)ethan-1-one
7-(2,2-dimethylpropyl)-2-[2-(4-methoxyphenyl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
N-(1-methyl-1H-1,2,3-triazol-4-yl)-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl 5-(cyclopentylamino)-1-(2-methoxyethyl)-3-(3-methylbutanamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-ethyl-4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]pyrimidine
1-methyl-6-oxo-N-(pyridin-3-ylmethyl)-N-(thiophen-3-ylmethyl)-1,6-dihydropyridine-3-carboxamide
1-butyl-4-[2-oxo-1-phenyl-2-(thiomorpholin-4-yl)ethyl]piperazine-2,3-dione
5-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-benzyl-3-{[(2-methoxyethyl)(methyl)amino]methyl}-N-methylimidazo[1,2-a]pyridine-2-carboxamide
methyl 2-{[8-(cyclopropylmethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]methyl}-1,3-oxazole-4-carboxylate
1-(1-{[3-(trifluoromethyl)phenyl]methyl}azetidin-3-yl)piperidine
6-[(diethylamino)methyl]-N-(1,4-dioxan-2-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
4-methyl-3-[(E)-2-phenylethenyl]benzamide
(3S)-1-{2-[(4-chlorophenyl)methyl]-1,3-benzoxazole-5-carbonyl}pyrrolidin-3-ol
(1S,5R)-3-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
6-(2,5-dimethylfuran-3-yl)-7-methyl-8-oxo-N-[(2R)-pyrrolidin-2-ylmethyl]-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-4-methyl-1,2,5-oxadiazole-3-carboxamide
N-{[5-(2-acetylphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-chlorothiophene-2-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}butan-1-one
3-(1H-pyrazol-1-ylmethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]benzamide
9-[(1S,3R)-3-aminocyclopentanecarbonyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(6-hydroxypyrimidin-4-yl)piperidin-1-yl]-4-(piperidin-1-yl)butan-1-one
2-[4-(1H-imidazol-2-yl)piperidin-1-yl]-N-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
N-cyclobutyl-3-{[3-(2-hydroxyethyl)-4-methylpiperazin-1-yl]sulfonyl}benzamide
2-[3-(dimethylamino)pyrrolidin-1-yl]-N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]acetamide
1-{2-[1-(2-chloro-5-fluorobenzoyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
ethyl 1-[5-(methoxymethyl)furan-2-carbonyl]-3-(3-phenylpropyl)piperidine-3-carboxylate
1-cyclopropanecarbonyl-4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]piperidine
5-(3-methoxyphenoxymethyl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,2-oxazole-3-carboxamide
1-[(3R,4R)-3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-(1,4-dioxan-2-ylmethyl)-5-ethyl-N,2-dimethylpyrimidin-4-amine
(3S,4R)-1-(1,3-benzoxazol-2-yl)-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[(1R,3R)-3-aminocyclopentyl]-3-(3-fluorophenyl)benzamide
5-(3-fluorophenoxymethyl)-N-methyl-N-[1-(3-methyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide