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1-(1-benzofuran-2-ylmethyl)-N-[3-(furan-2-yl)phenyl]piperidine-4-carboxamide
4-[1-(2,2-dimethylpropyl)pyrrolidin-3-yl]-1-(furan-3-carbonyl)piperidine
4-(1H-pyrazol-1-yl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine-4-carboxylic acid
methyl N-{2-[(3S,4R)-3-acetamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}carbamate
ethyl 4-{[4-(2,3-dihydro-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperazine-1-carboxylate
N-(3-chloro-2-ethoxyphenyl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
5-(3-methoxyphenoxymethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
1-(furan-3-ylmethyl)-N-[4-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
1-[1-(2-methyl-1-benzofuran-7-carbonyl)piperidin-4-yl]piperidin-3-ol
5-{1-[(2E)-3-(3-fluorophenyl)prop-2-enoyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
(2S)-3-(4-hydroxyphenyl)-2-{[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]formamido}propanoic acid
[3-(2-methoxyethyl)-1-{[6-(trifluoromethyl)pyridin-3-yl]methyl}piperidin-3-yl]methanol
N-(2-{1-[2-(1,3-thiazol-2-yl)ethyl]-1H-imidazol-2-yl}quinolin-6-yl)acetamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methyl-1-(1H-1,2,4-triazole-5-carbonyl)piperidine
2-[3-(1H-imidazol-1-yl)propyl]-9-(5-methyl-1,3-oxazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(2-aminoacetyl)-5-benzyl-1-(2-phenylphenyl)piperazin-2-one
3-[5-(2,3-dihydro-1-benzofuran-5-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(2,4-dimethoxyphenyl)ethan-1-one
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(methyl)[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amine
2-methyl-4-{[4-phenyl-5-(1-propyl-1H-imidazol-2-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazole
[(1-cyclohexylpiperidin-3-yl)methyl]({[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl})(pyridin-3-ylmethyl)amine
7-{4-[hydroxy(thiophen-2-yl)methyl]piperidine-1-carbonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-(oxan-2-ylmethyl)-4-phenyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-(3-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)benzonitrile
({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(4-phenylbutan-2-yl)amine
2-[(4-benzoylpiperazin-1-yl)methyl]-6-methylpyridin-3-ol
2-(morpholin-4-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
3-chloro-6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}pyridine-2-carboxylic acid
3-(1H-1,2,4-triazol-1-yl)-1-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}propan-1-one
N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-2-(pyridin-4-yl)pyrimidine-5-carboxamide
2,3,6-trimethyl-N-[2-(1,3-thiazol-4-yl)ethyl]quinoline-4-carboxamide
N-{[2-(dimethylamino)-8-methylquinolin-3-yl]methyl}-N-[2-(dimethylamino)ethyl]cyclohexanecarboxamide
2-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-N-methylpyridine-4-carboxamide
(1R,3S)-7-{[2-methoxy-5-(propan-2-yl)phenyl]methyl}-7-azaspiro[3.5]nonane-1,3-diol
4-(6-hydroxyhexyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
2-benzyl-8-(2,6-diaminopyrimidin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(2-hydroxyethyl)(methyl)amino]methyl}piperidin-2-one
3-(4-fluorophenyl)-N-[2-(oxan-2-yl)ethyl]propanamide
(1S,9S)-11-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-chloro-4-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
N-propyl-3-(pyridin-4-yl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-5-carboxamide
1-(4-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-({5-[3-(methylsulfanyl)butyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-2-{1H-pyrrolo[2,3-b]pyridin-1-yl}acetamide
5-{[(2-phenylethyl)(propan-2-yl)amino]methyl}pyrrolidin-2-one
(3R,4S)-1-(2,3-dimethoxybenzoyl)-4-(4-methoxyphenyl)pyrrolidin-3-amine
ethyl 3-[(2-fluorophenyl)methyl]-1-(furan-3-carbonyl)piperidine-3-carboxylate
{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}[(4-methoxyphenyl)methyl]amine
3-fluoro-N-{[7-(quinolin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}benzamide
6-(3-benzoylpiperidin-1-yl)-N-cyclopropyl-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine