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{7-fluoro-5-[4-(1H-imidazol-1-ylmethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
1-[4-(furan-2-yl)pyrimidin-2-yl]-N-[2-(4-methoxyphenyl)ethyl]-5-methyl-1H-pyrazole-4-carboxamide
1-(naphthalen-2-yl)-3-{2-[(2S)-pyrrolidin-2-yl]ethyl}urea
2-[(3-fluorophenyl)methyl]-4-(1,3-thiazol-2-ylmethyl)morpholine
1-{4-[3-(morpholine-4-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-(pyridin-3-yl)ethan-1-one
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2-oxo-1,2-dihydroquinoline-4-carboxamide
N,N-diethyl-2-({1-[(4-methoxyphenyl)methyl]-2-oxo-4-[2-(phenylsulfanyl)acetyl]-1,4-diazepan-6-yl}oxy)acetamide
1-[1'-(4-methylbenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
2-(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)-N-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]acetamide
(1S,2S)-N2-{1-[6-methyl-2-(propan-2-yl)pyrimidin-4-yl]piperidin-4-yl}-2,3-dihydro-1H-indene-1,2-diamine
2-methyl-4-(4-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}phenyl)butan-2-ol
1-[(2-chloro-4,5-dimethoxyphenyl)methyl]-4-[2-(methylsulfanyl)ethyl]piperazine
2,5-dimethyl-N-[3-(3-phenylpropanamido)phenyl]-1,3-oxazole-4-carboxamide
methyl 5-{[(4-fluorophenyl)methyl]amino}-3-(furan-2-amido)-1-(2-methoxyethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(3-methoxybenzoyl)piperazine
1-{imidazo[1,2-a]pyridine-6-carbonyl}-4-(thiophen-2-ylmethyl)-1,4-diazepane
4-({1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-4-ylmethyl)benzamide
2-[3-(pyridin-4-yl)-5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,4-triazol-1-yl]ethan-1-ol
N-cyclooctyl-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
N-(propan-2-yl)-4-({[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}amino)pyridine-2-carboxamide
3-(3-{[(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)amino]methyl}-1H-indol-1-yl)propanamide
1-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylpiperidine
2-(2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}phenoxy)ethan-1-ol
N-cyclopropyl-5-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-[4-(trifluoromethyl)pyrimidin-2-yl]pyrrolidin-3-yl]cyclobutanecarboxamide
2-(1H-1,3-benzodiazol-1-yl)-N-[2-(cyclohex-1-en-1-yl)ethyl]propanamide
N-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-4-(pyrimidin-2-yl)-1,4-diazepane-1-carboxamide
[(3R,4R)-4-[(4-methylpiperazin-1-yl)methyl]-1-[(4-phenyl-1,3-thiazol-2-yl)methyl]pyrrolidin-3-yl]methanol
1-cyclopentyl-4-(2,8-dimethylquinoline-4-carbonyl)piperazin-2-one
1-methyl-1'-(2-methyl-1-benzofuran-5-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
6-methyl-2-({4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)quinolin-4-ol
N-benzyl-2-[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
4-(4-fluorophenyl)-N-[2-(4-methyl-5-{[2-(morpholin-4-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]benzamide
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-2,6,8-trimethylquinoline-4-carboxamide
2-(5-acetylthiophen-3-yl)-N-[2-(2-methoxynaphthalen-1-yl)ethyl]acetamide
N-[(3-chloro-2,6-difluorophenyl)methyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
N-[4-(furan-2-yl)phenyl]-1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidine-3-carboxamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperazin-2-yl}ethan-1-ol
3-(hydroxymethyl)-1-[(5-methoxy-1H-indazol-3-yl)methyl]piperidin-3-ol
[(3R,4R)-1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
3-{2-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-methyl-6-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
N-(2-{[6-(2-methoxyphenyl)pyridazin-3-yl]amino}ethyl)acetamide
2-(adamantan-1-yl)-1-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}ethan-1-one
7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-4-[(5-methylfuran-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[(cyclopropylmethyl)(propyl)amino]-1-ethyl-N-(furan-3-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(3R,4R)-3-hydroxy-1-(3-methoxy-5-methylthiophene-2-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
3-ethyl-1-[3-(2-methoxyphenyl)propanoyl]piperidine-3-carboxylic acid
3-(2-methoxyethyl)-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
1-(2,2-dimethylpropyl)-4-{[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]amino}pyrrolidin-2-one