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2-(4-{[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-4-chloro-N-methylaniline
N-[(2R,3R)-2-(2-methoxyethoxy)-1'-(thiophene-3-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-methylpropanamide
(2R,3R,6R)-5-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[2-({[2-(dimethylamino)ethyl]amino}methyl)-5-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
(1R,5R)-6-(cyclobutylmethyl)-3-(1H-1,2,4-triazole-5-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}pyrrolidin-3-ol
N-[(3S,4S)-4-methoxypyrrolidin-3-yl]-2,6-dimethylquinoline-4-carboxamide
1-cyclopentyl-N-ethyl-6-oxo-N-(pyridin-4-ylmethyl)piperidine-3-carboxamide
(4aS,7aR)-6,6-dioxo-N-propyl-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
methyl({[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl})[3-(oxolan-2-yl)propyl]amine
2-(1H-indol-2-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
7-[(2,3-difluorophenyl)methyl]-2-[(1,2-dimethyl-1H-imidazol-5-yl)methyl]-2,7-diazaspiro[4.5]decane
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2,3-dihydro-1H-inden-2-amine
2-(cyclopropylmethyl)-4-oxo-N-(2-oxo-2,3-dihydro-1H-indol-5-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carboxamide
2-(2-ethyl-1H-imidazol-1-yl)-1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethan-1-one
1-cyclopentyl-4-{[3-(2,4-difluorophenyl)-1H-pyrazol-4-yl]methyl}piperazin-2-one
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-2-(2,3,6-trimethylphenoxy)acetamide
[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl](methyl){[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}amine
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-N-(pyridin-3-ylmethyl)-1-azabicyclo[2.2.2]octan-3-amine
2-(2-hydroxyethyl)-8-(2-methylpyridin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
[(5-{1-[(3-chloro-4-fluorophenyl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
3-chloro-N,6-dimethyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrazolo[1,5-a]pyrimidine-2-carboxamide
3-{2-carbamoyl-1-methyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-6-carbonyl}piperidine-1-carboxamide
(3S,4S)-1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3,4-diol
1-(3-{[3-(dimethylamino)pyrrolidin-1-yl]sulfonyl}benzoyl)piperidine-4-carbonitrile
1-(2-{1-[2-(4-chlorophenyl)-2-hydroxyacetyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
N-(2-{[3-(2-methylpropyl)-1,2-oxazol-5-yl]formamido}ethyl)pyridine-3-carboxamide
(2R,6R)-4-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(azepane-1-carbonyl)-N-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-chloro-4-{[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]methyl}phenol
propyl N-{[(3S,4S)-3-hydroxy-1-(3-hydroxypyridine-2-carbonyl)piperidin-4-yl]methyl}carbamate
2-{1'-[3-(furan-2-yl)propanoyl]-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl}acetamide
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]furan-2-carboxamide
1-cyclohexyl-N3-methyl-N5-[(2-methylphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-[5-methyl-4-(1-methyl-1H-pyrazol-4-yl)-1H-imidazol-2-yl]-1-(prop-2-en-1-yl)pyrrolidin-2-one
methyl 3-[(3S,4R)-1-[(2-hydroxyphenyl)methyl]-4-(pyrrolidin-1-yl)piperidin-3-yl]propanoate
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethan-1-one
2-cyclopentyl-9-(2-phenylbutanoyl)-2,9-diazaspiro[5.5]undecan-3-one
8-methoxy-3-[1-(thiophen-3-yl)propan-2-yl]-3,4-dihydroquinazolin-4-one
N,N-dimethyl-2-[4-(thiophen-3-yl)phenyl]acetamide
2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]acetamide
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
7-(2,3-dichlorobenzoyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(3-methoxybenzoyl)piperazine
(2S)-2-(dipropylamino)-N-(2,4,6-trimethylpyridin-3-yl)propanamide
6-(4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)pyridine-2-carbonitrile
N-cyclopropyl-N-({3-[(1-methylpiperidin-3-yl)methoxy]phenyl}methyl)pyridine-3-carboxamide
1,3-dimethyl-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)-1H-pyrazole-4-carboxamide
2,3-dimethoxy-N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]benzamide