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4-methyl-2-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-6-(trifluoromethyl)pyrimidine
(2R,3R)-3-(dimethylamino)-1'-(1,4-dithiepan-6-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]thiomorpholine
4-(2-methoxyphenoxy)-1-(trimethylpyrimidin-4-yl)piperidine-4-carboxylic acid
(3aR,6aR)-2-(azepane-1-sulfonyl)-5-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-5,6-dimethoxy-1,2-dihydroisoquinolin-1-one
3-(but-2-yn-1-yl)-5-{1-[(2-hydroxynaphthalen-1-yl)methyl]piperidin-4-yl}-5-(2-phenylethyl)imidazolidine-2,4-dione
N-[(3S,4R)-1-(4-aminopyrimidin-2-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
5-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]-1-(2-methylpropyl)-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
(2S,4S)-N-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-5-yl}-1-[(3-chlorophenyl)methyl]-4-(pyrimidin-2-ylsulfanyl)pyrrolidine-2-carboxamide
5-{2-[1-butyl-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-4,6-dimethylpyrimidin-2-ol
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-(methoxymethyl)-N-methylcyclobutane-1-carboxamide
3-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-{1-[(2-fluorophenyl)methyl]-1H-pyrazol-4-yl}urea
3-(3-fluorophenyl)-6-[(4-hydroxy-3-methoxyphenyl)methyl]-1-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
2-[(5-methylpyrazin-2-yl)methyl]-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-(cyclohexylmethyl)-N3,N3,N5-trimethyl-N5-[2-(4-methylphenoxy)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N,2-dimethyl-N-[(1-methylpyrrolidin-2-yl)methyl]-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
2-{2-[1-(3,6-dimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
(3R,4R)-3-cyclopropyl-4-methyl-1-[4-(methylamino)pyrimidin-2-yl]pyrrolidin-3-ol
2-acetyl-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-(isoquinolin-5-ylmethyl)-N,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
1-[2-({[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}amino)ethyl]imidazolidin-2-one
[5-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)furan-2-yl]methanol
1-benzoyl-4-[(2E)-2-methylpent-2-en-1-yl]piperazine
methyl 2-chloro-5-({[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]carbamoyl}amino)benzoate
2-(2,5-dioxoimidazolidin-1-yl)-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)acetamide
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]piperidin-4-amine
6-methoxy-3-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)quinolin-2-ol
N-ethyl-N-[(1-ethylpyrrolidin-3-yl)methyl]-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3-chlorophenyl)methyl]-4-[1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]piperazine
4-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-N,N-dimethylpiperazine-1-sulfonamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(oxane-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(4aR,7aS)-4-[(3,4-difluorophenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[2-(1-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
N-[(2,3-difluorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
3-(benzylsulfanyl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-(2-methoxyphenyl)-5-(1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-imidazol-2-yl)-1,3-thiazole
5-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
[3-(2-phenoxyethyl)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidin-3-yl]methanol
3-acetyl-N-(pyridin-3-ylmethyl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazole-5-carboxamide
methyl 3-acetamido-1-(3-methylbutyl)-5-[(oxan-4-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
1-[2-methoxy-4-(1,4-oxazepan-4-ylmethyl)phenoxy]-3-(pyrrolidin-1-yl)propan-2-ol
3-methyl-5-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)pyridine
5-methoxy-3-methyl-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
methyl 3-(1-acetylpiperidin-4-yl)-9-[2-(2-fluorophenyl)ethoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
3-(1H-1,3-benzodiazol-2-yl)-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)propanamide
N-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-(3-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-8-methylimidazo[1,2-a]pyridine-2-carbonyl)morpholine
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]benzamide