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3-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-1,3-oxazolidin-2-one
3-cyclohexyl-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]-1H-pyrazole-4-carboxamide
2-[(4-methoxyphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-1,3-benzoxazole
(4aR,7aS)-1-propyl-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-[4-(trifluoromethyl)pyrimidin-2-yl]-2,7-diazaspiro[4.4]nonane-1,3-dione
1-[(3-fluorophenyl)methyl]-4-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazine
1-(4-{[(6-methoxy-1,3-benzothiazol-2-yl)amino]methyl}thiophen-2-yl)ethan-1-one
2-[(4-chlorophenyl)methyl]-8-[2-(2-methoxyethoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
2-methoxy-N-(1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
2-[(3-methoxyphenyl)methyl]-4-(pyridin-3-ylmethyl)morpholine
N-(1-{2-[4-(3,5-dimethylphenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-4-oxo-4-phenylbutanamide
1-(4-hydroxy-2-methylpyrimidine-5-carbonyl)-4-phenylpiperidine-4-carbonitrile
1-(2-hydroxy-3-methoxybenzoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
7-(1,3-benzothiazol-2-yl)-4-[(5-chlorothiophen-2-yl)sulfonyl]-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[(4-fluorophenyl)methyl]piperidine
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-methyl-N-(quinolin-8-ylmethyl)acetamide
N-methyl-N-(oxan-2-ylmethyl)-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
7-fluoro-3-methyl-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]-1H-indole-2-carboxamide
3-[1-(2,6-dimethylpyridin-4-yl)-N-(2-phenylethyl)formamido]propanamide
N-{2-[1-(2,3,4-trifluorobenzenesulfonyl)piperidin-2-yl]ethyl}acetamide
6-[2-(2-methylpyrimidin-5-yl)-1H-imidazol-1-yl]quinoline
2-{2,5-dioxo-3-phenyl-1-[3-(pyridin-3-yloxy)propyl]pyrrolidin-3-yl}-N-(1H-imidazol-2-ylmethyl)-N-methylacetamide
N-(1,1-dioxo-1λ6-thian-4-yl)-1-(furan-2-ylmethyl)-N-methylpiperidine-3-carboxamide
2-(4-fluorophenyl)-4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)morpholine
N-methyl-3-[2-(naphthalen-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)propanamide
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-methylprop-2-en-1-yl)benzamide
2-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)ethan-1-ol
2-amino-4-[4-(1H-pyrazol-1-ylmethyl)phenyl]-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
4-(2-chloro-4-fluorophenyl)-3,6-dimethyl-[1,2]oxazolo[5,4-d]pyrimidine
8-[(1R,3S)-3-aminocyclohexanecarbonyl]-3-hexyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(3S,4R)-3-carboxy-4-(2-methylphenyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
9-[(4-methoxypyridin-2-yl)methyl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aR)-5-(2-aminopyridine-4-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
1-cyclohexyl-N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethylpiperidine-4-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(oxolan-2-ylmethyl)-2-{3-[3-(1,3-thiazol-2-yl)phenyl]-1H-pyrazol-1-yl}acetamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-2-(phenylamino)pyrimidine-5-carboxamide
4-[7-(6-cyanopyridin-2-yl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
6-ethyl-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-methyl-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}-N-(pyrazin-2-ylmethyl)acetamide
1,N3-dibenzyl-N3-methyl-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
[1-(5-chloro-3-phenyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methanamine
1-(methoxymethyl)-N-{2-[3-(trifluoromethyl)phenyl]ethyl}cyclopropane-1-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-N-methyl-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)acetamide
1-(1H-pyrazole-4-carbonyl)-4-(pyridin-3-yl)piperazine
4-{1-[1-(3-methoxypyrazin-2-yl)piperidin-4-yl]ethyl}morpholine
N-[(3-chlorophenyl)methyl]-2-(3-methoxyphenoxymethyl)-N-methyl-1,3-oxazole-4-carboxamide
2-(3-tert-butyl-5-{spiro[2.3]hexan-1-yl}-1H-1,2,4-triazol-1-yl)ethan-1-ol
3-(3,4-dimethylphenyl)-1-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]propan-1-one
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-5-methyl-1,3,4-oxadiazole-2-carboxamide