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N-[(2-aminopyrimidin-5-yl)methyl]-N-methyl-2-[4-(pyrrolidine-1-carbonyl)morpholin-3-yl]acetamide
2-{N-[(2-methoxyphenyl)methyl]-1-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]formamido}acetic acid
N-{[2-(azocan-1-yl)pyridin-3-yl]methyl}-3-(3-methyl-1H-pyrazol-1-yl)propanamide
2-[3-(1-methyl-1H-1,2,4-triazol-5-yl)-1H-pyrazol-1-yl]-N-[1-methyl-3-(propan-2-yl)-1H-pyrazol-5-yl]acetamide
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N,6-dimethylpyrimidin-2-amine
1-methyl-1'-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
4-methyl-5-{1-[3-(trifluoromethyl)phenyl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,3-oxazole
{[2-(azepane-1-carbonyl)-7-methylimidazo[1,2-a]pyridin-3-yl]methyl}[1-(4-methoxyphenyl)ethyl]methylamine
1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}azepane
N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-3,5-dimethyl-1,2-oxazole-4-sulfonamide
1-cyclohexyl-4-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperazine
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-N-(2-methoxyethyl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
4-{[methyl(thian-4-yl)carbamoyl]amino}-N-(oxolan-2-ylmethyl)benzamide
4-methyl-7-(methylsulfanyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinolin-2-amine
1-(cyclopropylmethyl)-5-{8-methylimidazo[1,2-a]pyridine-2-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
1-[2-methoxy-4-({[2-(6-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-cyclohexyl-5-(methoxymethyl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
2-[(4-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-1-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-2-yl}ethan-1-one
1-cyclobutyl-3-[2-(methylsulfanyl)benzoyl]piperidine
3-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-N-(4-methoxyphenyl)benzamide
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methoxyethyl)-3-(2-methylpropyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3S,4S)-1-(1-benzylpiperidin-4-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-2,8-diazaspiro[4.5]decane-3-carboxamide
1-[1-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-2-phenylethan-1-ol
1'-(2-methoxypyridine-4-carbonyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
8-chloro-2-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazol-4-yl}quinoline
3-[(2S,4S)-2-{[(dimethylsulfamoyl)amino]methyl}-4-fluoropyrrolidine-1-carbonyl]-N,N-dimethylaniline
N-[1-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
1-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]phenyl}imidazolidine-2,4-dione
3-[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]-6-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-[2-(dimethylamino)-2-(5-methylfuran-2-yl)ethyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide
ethyl 3-{[3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}propanoate
1-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-3-(4-methyl-4H-1,2,4-triazol-3-yl)propan-1-one
N-[(2,3-difluorophenyl)methyl]-1-(4,7-dimethylquinazolin-2-yl)piperidine-4-carboxamide
3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-1-(2-methoxyethyl)-3-(2-methoxyphenyl)pyrrolidine-2,5-dione
N-[(3R,4R)-3-hydroxy-1-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]piperidin-4-yl]pyridine-2-carboxamide
5-{3-[benzyl(methyl)amino]piperidine-1-carbonyl}-2,1,3-benzoxadiazol-1-ium-1-olate
4-({4-[(3,5-dimethylphenyl)methyl]-3-oxopiperazin-1-yl}methyl)-1-ethyl-1H-pyrrole-2-carbonitrile
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methyl-6-(piperidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
4-(6-chloro-1,3-benzothiazol-2-yl)-N,N-dimethylbenzamide
methyl (2S,4S,5R)-4-[ethyl(methyl)carbamoyl]-1-methyl-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylate
N-methyl-3-(propan-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-4,5-dihydro-1,2-oxazole-5-carboxamide
(1R,7S)-3-(3-methylbutyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(2S)-3-(4-hydroxyphenyl)-2-[(3-propyl-1H-pyrazol-5-yl)formamido]propanoic acid
N-{4-[(2S)-2-hydroxy-3-phenylpropanamido]phenyl}pentanamide
N-[(2,5-dimethoxyphenyl)methyl]-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
{[4-(3-chlorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}[(2,5-dimethylphenyl)methyl]methylamine
N-[2-(azepan-1-yl)ethyl]-3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-(propan-2-yl)propanamide
N-[(1-acetylpiperidin-3-yl)methyl]-3-(4-methoxyphenyl)prop-2-ynamide