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N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-(methylsulfanyl)pyridine-3-carboxamide
5-methyl-N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1,2-oxazole-4-sulfonamide
2-[2-(methylsulfanyl)phenyl]-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(3S)-2-oxoazepan-3-yl]propanamide
2-(3-chloro-4-hydroxyphenyl)-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]acetamide
(2S)-1-[2-(1H-imidazol-4-yl)acetyl]-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
(3S,4S)-1-(3,5-dichloro-2-methoxybenzoyl)piperidine-3,4-diol
3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-(oxolan-3-yl)-3-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
4-(2-{4-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperazin-1-yl}ethyl)morpholine
2-(2-methoxy-4-methylphenoxymethyl)-N-(1,2-oxazol-3-ylmethyl)-1,3-oxazole-4-carboxamide
3-methoxy-N-{1-[7-({4-[methyl(phenyl)amino]phenyl}methyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}propanamide
(4aS,7aR)-1-(5-chloropyridine-2-carbonyl)-4-cyclopropanecarbonyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-cyclobutyl-9-[(2S)-3-hydroxy-2-(methylamino)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{6-[(1E)-pent-1-en-1-yl]pyrazine-2-carbonyl}morpholine
4-{3-[(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)oxy]benzoyl}morpholine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-5-phenyl-1,2-oxazole-3-carboxamide
2-(4-{[3-(hydroxymethyl)-4-(propan-2-yloxy)phenyl]methyl}-1-(propan-2-yl)piperazin-2-yl)ethan-1-ol
N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
8-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-hydroxy-2-(pyridin-3-yl)-N-[2-(pyridin-4-yl)ethyl]pyrimidine-5-carboxamide
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]acetamide
2-methoxyethyl N-{[(3S,4S)-1-cycloheptyl-3-hydroxypiperidin-4-yl]methyl}carbamate
(4aR,8aR)-4-[4-(piperidin-1-ylmethyl)benzoyl]-octahydro-2H-1,4-benzoxazine
7-fluoro-N-{2-[3-(2-methylphenyl)pyrrolidin-1-yl]ethyl}quinazolin-4-amine
1-{1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
3-(3-chloro-1,2-oxazol-5-yl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}propanamide
2-[(3,4-difluorophenyl)methyl]-8-[3-(methylsulfanyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[1-(7-{[5-(hydroxymethyl)furan-2-yl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)-3-methylbutyl]-3,5-dimethylbenzamide
5-[(3-hydroxyphenyl)methyl]-N-(2-methoxyethyl)-1-(3-methylbutyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-methyl-N-(1-{1-[5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carbonyl]piperidin-4-yl}-1H-pyrazol-5-yl)butanamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(6-methoxy-2-oxo-2,3-dihydro-1H-indol-3-yl)acetamide
2-{4-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]piperidin-1-yl}-4,6-dimethylquinazoline
5-(2-chlorophenyl)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]furan-2-carboxamide
2-cyclopropyl-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]pyrimidin-4-ol
1-[(5-chloro-2,4-dimethoxyphenyl)methyl]-4,4-difluoropiperidine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
2,8-dimethyl-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]quinoline-4-carboxamide
N-({4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-2-(pyridin-2-ylsulfanyl)acetamide
1-(carbamoylmethyl)-N-[3-(2-hydroxyphenyl)propyl]piperidine-3-carboxamide
N-methyl-3-(1-methylpiperidin-3-yl)-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)propanamide
2-chloro-5-acetamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
6-{[2-(trifluoromethyl)phenyl]methyl}-5,6-dihydro-1,6-naphthyridin-5-one
(1R,2R,6S,7S)-N-[4-(furan-2-ylmethoxy)phenyl]-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
4-acetyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]benzamide