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1-{1-[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}propan-1-ol
N-cyclopropyl-5-(2-oxopentanoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
4-[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-1-phenylpiperazin-2-one
1-(4-ethylpiperazin-1-yl)-3-(2-methoxy-4-{[(2-methoxyethyl)amino]methyl}phenoxy)propan-2-ol
4-{1-[6-(2-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]piperidin-4-yl}thiomorpholine
4-(2,6-dimethylpyridin-3-yl)-N-[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]pyrimidin-2-amine
N-[(4-benzyl-5-{[(2-chlorophenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]-2-(2-methyl-1,3-thiazol-4-yl)acetamide
N-(3-chloro-4-methylphenyl)-3-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-3-oxopropanamide
N-({1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl}methyl)-4H-thieno[3,2-b]pyrrole-5-carboxamide
9-[(3,5-dimethyl-4-oxo-1,4-dihydropyridin-2-yl)methyl]-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(dimethylamino)-7-(methylsulfanyl)quinolin-3-yl]methyl}-3-fluoro-N-(3-methoxypropyl)benzamide
N3-[6-(methoxymethyl)pyrimidin-4-yl]-N1-(pyridin-3-yl)propane-1,3-diamine
N-methyl-5-[(2-methylpropyl)amino]-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
2-{4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-N,N-dimethylacetamide
N-[4-(isoquinolin-5-yl)-6-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]-2-methylpropanamide
(1S,4S)-2-(5-chloro-2-methoxyphenyl)-5-[1-(2-phenylethyl)piperidin-4-yl]-2,5-diazabicyclo[2.2.1]heptan-3-one
5-(2-ethylpiperidine-1-carbonyl)-N-(furan-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
3-[2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
3-{5-[(3-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}-1-[2-(1H-pyrazol-4-yl)ethyl]urea
N-(2,6-dimethylphenyl)-3-[2-(2-ethyl-1H-imidazol-1-yl)acetamido]benzamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)acetamide
3-(dimethylsulfamoyl)-N-[(1R)-1-(4-methoxyphenyl)ethyl]-5-({[3-(trifluoromethyl)phenyl]methyl}amino)benzamide
6-(2H-1,3-benzodioxol-5-yl)-1H-1,3-benzodiazole
7-(oxan-4-yl)-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-({4-[4-(3-methoxyphenyl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyridine
6-[1-(morpholin-4-yl)cyclohexanecarbonyl]-N-[2-(pyridin-2-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
4-ethanesulfonamido-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
N-(2-methanesulfonamidoethyl)-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
({3-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]pyrazolo[1,5-a]pyrimidin-6-yl}methyl)diethylamine
4-amino-1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]butan-1-one
[(5-{[2-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}thiophen-3-yl)methyl]dimethylamine
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methyloxetan-3-yl)methyl]amine
1-(2,2-dimethylpropyl)-3-{[(2,2-dimethylpropyl)amino]methyl}-3-hydroxypiperidin-2-one
ethyl 1-benzyl-5-[3-(3-hydroxy-3-methylbut-1-yn-1-yl)benzoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-ethyl-1-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methyl)urea
N-(2-{7-[(2-methoxynaphthalen-1-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-4-methylbenzamide
N-[2-(4-methoxyphenyl)phenyl]-1-[(2-methyl-1H-imidazol-4-yl)methyl]piperidine-3-carboxamide
4-(1-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]piperidin-4-yl}piperidine-3-carbonyl)morpholine
[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]({[2-(propylsulfanyl)pyrimidin-5-yl]methyl})amine
2-(1H-indol-3-yl)-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-(3-methyl-1,2,4-thiadiazol-5-yl)-4-azaspiro[2.5]octane-4-carboxamide
[1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(pyrazin-2-yl)piperidin-3-ol
2-{1-methyl-4-[(3-phenoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
3-[3-(dimethylamino)propyl]-5-[(4-fluorophenyl)methyl]-5-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)imidazolidine-2,4-dione
3-chloro-5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1,2-dihydropyridin-2-one
1-{6-hydroxy-4-[2-(morpholin-4-yl)benzoyl]-1,4-diazepan-1-yl}ethan-1-one
N,N-dimethyl-1-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]pyrrolidin-3-amine
2-{4-[(5-methylfuran-2-yl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
6-methoxy-3-{[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]methyl}-1H-indazole