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8-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[3-(dimethylamino)propyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl (2S)-2-({5-[(2-methoxyethyl)carbamoyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridin-3-yl}formamido)-2-phenylacetate
5-(2,3-difluoro-6-methoxyphenyl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-4-phenyl-1H-imidazole
N-(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
(1-{5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperidin-2-yl)methanol
5-[(3aS,6aS)-1-[(4-fluoro-3-methylphenyl)methyl]-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2-ethyl-4-methyl-1,3-oxazole
1-{5-acetyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-phenylethane-1,2-dione
5-[(isoquinolin-5-yloxy)methyl]-N-[1-(pyridin-3-yl)propan-2-yl]-1,2-oxazole-3-carboxamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-[(4-chlorophenyl)methyl]-4-{[(3,4-difluorophenyl)methyl]amino}pyrrolidine-2-carboxamide
3-methyl-N-[1-(pyrimidin-2-yl)piperidin-3-yl]thiophene-2-carboxamide
N-[1-(2-methoxyphenyl)-5-oxopyrrolidin-3-yl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-(2-methoxyethyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
8-[(2R)-2-aminopropanoyl]-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(2R,3R)-3-amino-1'-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
3-(4-methanesulfonyl-1,4-diazepane-1-carbonyl)-2-methyl-1,2,3,4-tetrahydroisoquinoline
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[2-(1H-imidazol-4-yl)ethyl]-1-(2-methylpropyl)piperidine-3-carboxamide
methyl[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl][(2-methyl-1H-imidazol-4-yl)methyl]amine
(1S,5R)-6-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-[(3S,4R)-3-hydroxy-4-(3-methylthiophen-2-yl)piperidin-1-yl]-3-(2-methoxyphenyl)propan-1-one
1-[(1-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}piperidin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxylic acid
2-amino-N-[2-(4-acetamidophenyl)phenyl]acetamide
2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-(2-hydroxypropyl)-5-methoxybenzamide
6-{3-[1-(2,5-difluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
(4aR,7aS)-1-ethyl-4-(pyrrolidine-1-sulfonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-(4-methoxyphenyl)-2-{1-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-imidazol-2-yl}-1H-imidazole
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
N-[2-(1,3-thiazol-2-yl)ethyl]-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]-3-(1H-pyrazol-1-ylmethyl)benzamide
methyl (2S)-1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carboxylate
5-methoxy-N-(6-methoxy-1,2,3,4-tetrahydronaphthalen-1-yl)-1-methyl-1H-indole-2-carboxamide
3-[(3R,4S)-1-[(1-methyl-1H-indol-2-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
2-[4-(2,1,3-benzoxadiazol-4-ylmethyl)-1-[(2-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-(2-{[(4-chlorophenyl)methyl](methyl)amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
1-[(3-chlorophenyl)methyl]-5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)azepan-2-one
3-[(3-acetyl-1H-pyrazol-5-yl)formamido]-N-cyclohexylpropanamide
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-(1,3-thiazol-2-ylmethyl)pyridin-2-amine
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-4-yl}propanamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-5-(pyrrolidine-1-carbonyl)pyridin-2-amine
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-4-carboxamide
3-[3-(3-hydroxy-3-methylbutyl)benzoyl]-3,9-diazaspiro[5.6]dodecan-10-one
2-(hydroxymethyl)-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-1-carboxamide
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-3-(2-methoxyphenyl)-1-methylpyrrolidine-2,5-dione
2-({5-[(4-hydroxyphenyl)methyl]-4-(1-phenylethyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
6-{[5-oxo-1-(3-phenylpropyl)pyrrolidin-3-yl]amino}pyridine-2-carbonitrile
1-(but-3-enoyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
2-methoxy-5-({3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzoic acid
{[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}[(1-methyl-1H-pyrazol-4-yl)methyl]amine
8-methyl-3-{[4-(morpholin-4-yl)piperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
6-[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one