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N-methyl-N-[(4-methylphenyl)methyl]-4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzamide
N,2,6-trimethyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]quinoline-4-carboxamide
N-cyclohexyl-2-[1-cyclopentyl-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-(prop-2-yn-1-yl)acetamide
3-[(3S,4R)-1-[(4-chlorophenyl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]-N-[3-(dimethylamino)propyl]propanamide
methyl 2-[1-benzyl-8-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(3aS,7aR)-5-methyl-2-(5-methyl-1,3,4-thiadiazol-2-yl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-(2-chlorophenyl)-4-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)pyrrolidin-2-one
N-methyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-oxazolidine-4-carboxamide
methyl 1-methoxy-2-oxo-8-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
5,6-dimethyl-N-[3-(pyridin-3-yl)propyl]thieno[2,3-d]pyrimidin-4-amine
2-amino-4-(4-methoxy-2-methylphenyl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
3-ethoxy-N-[(3R,4S)-1-[4-(methylamino)pyrimidin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]propanamide
5-{[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N,N-dimethylfuran-2-carboxamide
3-[5-(2-methyl-3-phenylcycloprop-2-en-1-yl)-1,2,4-oxadiazol-3-yl]pyridazine
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(furan-2-yl)ethyl]acetamide
3-(hydroxymethyl)-1-({1-[(4-methylphenyl)methyl]-1H-1,3-benzodiazol-2-yl}methyl)piperidin-3-ol
1-(dimethyl-1,3-oxazole-4-carbonyl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
5-(dimethylamino)-2-{[2-(2-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
N-[1-(2-fluorophenyl)piperidin-4-yl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-methyl-N-(1-{1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]piperidin-4-yl}-2-phenylethyl)-2-(1H-pyrazol-1-yl)acetamide
N-[(1-ethylpiperidin-3-yl)methyl]-1-propyl-1H-pyrazole-5-carboxamide
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]thiophene-2-sulfonamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-cyclopentyl-1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-phenylethan-1-one
1-benzyl-2-methyl-3-[2-(1,2-oxazinan-2-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
(3aR,5S,6S,7aS)-2-(quinoxalin-2-yl)-octahydro-1H-isoindole-5,6-diol
1-(3-methoxypropanoyl)-N-[3-(3-methylphenyl)phenyl]piperidine-3-carboxamide
methyl 1-[(3S,5S)-5-{[2-(1H-indol-3-yl)ethyl]carbamoyl}-1-[(2-methoxyphenyl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[5-(2-methoxyacetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
3-{2-[2-(3-fluorophenyl)azepan-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
N-{[(2S,4S)-4-fluoro-1-(thiophene-3-carbonyl)pyrrolidin-2-yl]methyl}-2-phenoxyacetamide
1-(4-{[3-(3-hydroxypiperidine-1-carbonyl)-1,2-oxazol-5-yl]methoxy}phenyl)ethan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-cyclopropyl-5-[4-(morpholin-4-yl)piperidine-1-carbonyl]pyridin-2-amine
methyl 3-{[2-(3-methoxypropyl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]methyl}benzoate
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1H-indole-6-carboxamide
(1S,5R)-6-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
6-[4-(4-benzyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]pyridine-3-carboxamide
4,5-dimethyl-6-(3-phenylpiperazin-1-yl)pyrimidine
4-(2-methyl-1-benzofuran-5-carbonyl)thiomorpholine
4-(1-methyl-1H-imidazol-2-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
7-(3-chlorophenyl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-({9-ethyl-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}methyl)benzoic acid
1-[4-(2-hydroxyethyl)piperazin-1-yl]-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]propan-1-one
2-{4-[2-(benzyloxy)ethyl]-6-hydroxy-1,4-diazepan-1-yl}acetic acid
N-(2,2-dimethyloxan-4-yl)-N-ethyl-3-(3-hydroxy-3-methylbutyl)benzamide
3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl]-7-methyl-1H-indole