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N-(3-hydroxypropyl)-N-methyl-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
6-(2,1,3-benzothiadiazol-5-ylmethyl)-N-(3,5-dimethylphenyl)-6-azaspiro[2.5]octane-1-carboxamide
methyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl){[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
N-benzyl-N,1-dimethyl-5-{methyl[2-(pyridin-2-yl)ethyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}imidazo[1,2-a]pyridine-6-carboxamide
2-[4-(2-amino-9H-purin-6-yl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
N-(1-{1-[(2-hydroxy-3-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
N-({1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}methyl)cyclobutanecarboxamide
1-cyclopropyl-5-oxo-N-[2-(1H-pyrrol-1-yl)ethyl]pyrrolidine-3-carboxamide
1-[(3R,4R)-4-amino-3-hydroxypiperidin-1-yl]-2-(9-methyl-9H-carbazol-3-yl)ethan-1-one
2,2-dimethyl-1-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one
2-{[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]methyl}-6-ethoxyphenol
(3R,4R)-1-[4-(4-fluorophenyl)oxane-4-carbonyl]-4-(hydroxymethyl)piperidin-3-ol
7-{[2-methyl-5-(1,2-oxazol-5-yl)thiophen-3-yl]sulfonyl}-2-oxa-7-azaspiro[4.5]decane
N-ethyl-N-[1-(4-methoxyphenyl)propan-2-yl]-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidine-2-carboxamide
2-{[2-(furan-2-yl)-7-(1H-imidazol-4-ylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
methyl 6-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-(thiomorpholine-4-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-benzyl-3-[1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)piperidin-4-yl]-N-methylpropanamide
N-(oxolan-3-yl)-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-[(3R,4S)-4-(morpholin-4-yl)-1-(quinolin-8-ylmethyl)piperidin-3-yl]propan-1-ol
2-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
5-({[3-(1H-imidazol-1-yl)propyl]amino}methyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
1,4-dimethyl-9-(1-methyl-1H-indazole-3-carbonyl)-1,4,9-triazaspiro[5.5]undecane
N-{[2-(4-methyl-1,4-diazepan-1-yl)pyridin-3-yl]methyl}piperidine-1-sulfonamide
3-[({4-benzyl-5-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}sulfanyl)methyl]pyridine
1-cyclohexyl-N-(oxolan-2-ylmethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N-(1-{7-[(4-hydroxy-2-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)pyridine-2-carboxamide
N-(1-{1-[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
4-({[1-(pyrrolidin-1-yl)cyclopentyl]methyl}amino)pyrimidine-5-carboxylic acid
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-{octahydropyrrolo[1,2-a]piperazin-2-yl}-3-phenoxypropan-1-one
ethyl 2-[2-(4-chlorophenyl)morpholin-4-yl]-1,3-oxazole-4-carboxylate
4-{1-[1-(pyrrolidin-1-yl)cyclopentanecarbonyl]piperidin-3-yl}benzoic acid
(2E)-1-{3-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]piperidin-1-yl}-2-methylbut-2-en-1-one
1-{4-[(3-fluorophenyl)methyl]-4-(hydroxymethyl)piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
(3S,4R)-1-(2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-[2-(4-chlorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-pyrazole
4-{1-[2-(propan-2-yloxy)acetyl]piperidin-3-yl}benzoic acid
2-(4-fluorophenoxymethyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1,3-oxazole-4-carboxamide
3-(4-chloro-2-methylbenzoyl)-1-cyclohexanecarbonylpiperidine
1-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)urea
2-{3-[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]phenyl}pyridine
(3S,9aR)-3-benzyl-8-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-(2-{[4-hydroxy-4-(pyrrolidin-1-ylmethyl)piperidin-1-yl]methyl}phenoxy)acetic acid
1-(piperidin-1-yl)-3-[2-({[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-propyl-4-[4-(1H-1,2,3,4-tetrazol-1-ylmethyl)benzoyl]morpholine
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amine
5-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-2-(propan-2-yl)pyrimidine