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2-(1,3-benzothiazol-2-ylmethyl)-4-{4-[4-(2,5-dimethylphenyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-(4-{[4-(2-methylphenyl)-1,4-diazepan-1-yl]methyl}phenyl)imidazolidin-2-one
N3-ethyl-N5-[(4-fluorophenyl)methyl]-1-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
4-(3-phenylpiperidin-1-yl)-6-(propan-2-yl)pyrimidine
2-(3-{[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
1-(1,3-benzoxazol-2-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]piperidin-4-amine
3-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-[2-(trifluoromethoxy)phenyl]urea
1-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-oxoethyl)-1,2-dihydroquinoxalin-2-one
1-[1'-(4-chlorobenzoyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
N-(cyclopropylmethyl)-1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-({3-[(2-methylpropyl)(thiophen-2-ylmethyl)carbamoyl]phenyl}amino)acetic acid
6-{4-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-N,N-dimethylpyridine-3-carboxamide
1-(2-methylpropyl)-4-(1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidin-3-yl)piperidine
methyl 1-(2-methoxyethyl)-2-oxo-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylate
1-(cyclopropylmethyl)-N-ethyl-5-[(1-methyl-1H-indol-3-yl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(2S,4R)-N-(2-methoxyethyl)-4-[(naphthalen-2-ylmethyl)amino]-1-(propan-2-yl)pyrrolidine-2-carboxamide
methyl 3-(3-methylbutyl)-7-oxo-9-[2-(pyridin-2-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-(3-fluoro-4-methylbenzoyl)-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
N-ethyl-2-{8-ethyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-4-carboxamide
3-(4-methoxy-4-phenylpiperidine-1-carbonyl)-2-methyl-2,8-diazaspiro[4.5]decane
1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(1H-1,2,4-triazole-3-carbonyl)piperazine
N,N-dimethyl-5-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyridin-2-amine
8-(2,2-dimethylpropyl)-1-ethyl-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-cyclopentyl-2-[2-(2-oxoazepan-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
3-{1-[(2-hydroxyphenyl)methyl]piperidin-4-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-{6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-cyclopropanecarbonylpiperidin-3-amine
1-{3-[(4-ethylpiperazin-1-yl)methyl]phenoxy}-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-2,3-dimethoxybenzamide
ethyl 4-(2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetyl)piperazine-1-carboxylate
N-(furan-2-ylmethyl)-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-(pyridin-4-ylmethyl)acetamide
2-tert-butyl-6-{furo[3,2-c]pyridin-4-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
7-(1-benzothiophen-3-yl)-9-methoxy-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-{[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)-1,4-diazepane
N-[2-(2-methoxy-5-{[4-(2-methylphenyl)piperazin-1-yl]methyl}phenoxy)ethyl]-3-methylthiophene-2-carboxamide
3-(2-fluoro-6-methoxyphenyl)-4-methylpyridine
9-[(2,4-diethoxy-3-methylphenyl)methyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
1-benzyl-2-methyl-3-{2-[(3R)-3-methylpiperazin-1-yl]-2-oxoethyl}-4,5,6,7-tetrahydro-1H-indol-4-one
1-{2-[(cyclohex-3-en-1-ylmethyl)amino]ethyl}-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
5-methoxy-N,1-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-indole-2-carboxamide
3-[(butylamino)methyl]-3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
{[1-(cyclohexylmethyl)-2-methanesulfonyl-1H-imidazol-5-yl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})methylamine
2-(2,5-dioxoimidazolidin-1-yl)-N-methyl-N-(quinoxalin-2-ylmethyl)acetamide
9-(2-hydroxybutanoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-5-[4-(1H-imidazol-1-yl)butanoyl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(furan-2-ylmethyl)-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-[2-(4-fluorophenyl)pyrrolidine-1-carbonyl]-4-methyl-2-(propan-2-yl)-1,3-thiazole
4-{3-[4-(4-chlorophenyl)-4-hydroxypiperidine-1-carbonyl]piperidin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
methyl 4-(5-methyl-4-{[methyl(oxolan-3-yl)amino]methyl}-1,3-oxazol-2-yl)benzoate
{2-[4-(2-methoxypyridine-4-carbonyl)morpholin-2-yl]ethyl}dimethylamine
1-[4-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one