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4-[(2,3-dimethoxyphenyl)methyl]-7-{[4-(4-fluorophenyl)piperazin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-{2-[(3-methylpyridin-4-yl)amino]ethyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(butan-2-yl)acetamide
N3-[2-(cyclohex-1-en-1-yl)ethyl]-N5-ethyl-1-[(2-methoxyphenyl)methyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
1-[6-(2-fluorophenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-3-(methoxymethyl)piperidine
5-(4-acetyl-4-phenylpiperidine-1-carbonyl)-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
5-(2-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethyl-1,2,5-oxadiazole-3-carboxamide
2,2-diethyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclopropane-1-carboxamide
3-{1-oxaspiro[4.4]nonan-3-yl}-1-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
N-cyclopropyl-2-[(1E)-pent-1-en-1-yl]pyridine-4-carboxamide
N-[(3R,4R)-4-(morpholin-4-yl)oxolan-3-yl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-({4-[(3-chlorophenyl)methyl]piperazin-1-yl}methyl)-6-fluoroquinolin-4-ol
5-{2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-3-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(prop-2-en-1-yl)(pyridin-2-ylmethyl)amine
N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-methylpyridin-2-amine
N-[(2R,3R)-2-ethoxy-1'-(1H-pyrazole-4-carbonyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]pyridine-3-carboxamide
methyl (2S,4R)-1-[(2,5-difluorophenyl)methyl]-4-(2,3-dimethyl-1H-indole-7-amido)pyrrolidine-2-carboxylate
2-{[(4-acetylphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
1-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}cyclobutane-1-carboxamide
(1R,5S,8S)-8-methoxy-3-{2-methylthieno[2,3-d]pyrimidin-4-yl}-3-azabicyclo[3.2.1]octane
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[(3,5-difluorophenyl)methyl]pyrrolidin-2-one
4-[2-(3,4-dimethoxyphenyl)acetyl]-1-(2-methylphenyl)piperazin-2-one
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[2-hydroxy-3-(4-{[(1H-indol-4-ylmethyl)amino]methyl}-2-methoxyphenoxy)propyl]piperidin-4-ol
(2Z)-N-({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)-3-(3,4-dimethoxyphenyl)prop-2-enamide
4-(cyclopentylmethyl)-1-(4-methoxyphenyl)piperazin-2-one
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-[(3-hydroxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
1-methyl-2-(2-{3-[4-(trifluoromethyl)phenyl]-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethyl)pyrrolidine
2-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-2,3-dihydro-1H-isoindole
N-[(2R,3R)-1'-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-2-(prop-2-en-1-yloxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(methylamino)pyridine-3-carboxamide
1-(dimethylamino)-3-(4-methoxy-2-{[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]methyl}phenoxy)propan-2-ol
4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-yl}-7-methylthieno[3,2-d]pyrimidine
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
1-benzyl-N5-cyclopropyl-N3-methyl-4-oxo-N3-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
2-({3-[4-(2,6-difluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-5-methoxyphenol
1-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-3-(2-methylphenyl)pyrrolidin-3-ol
2-(4-{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
2-{[1-methyl-3-(2-methylpropyl)-1H-pyrazol-5-yl]formamido}-N-(1,3-thiazol-2-yl)acetamide
4-methyl-5-[3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrimidine
N-(2H-1,3-benzodioxol-5-ylmethyl)-2-(5-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1H-1,2,3,4-tetrazol-1-yl)acetamide
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-1-[3-(3-ethylphenoxy)azetidin-1-yl]propan-1-one
N-[3-(4-fluorophenyl)propyl]-2-oxo-1-oxaspiro[4.4]nonane-4-carboxamide
(1R,5R)-6-(cyclobutylmethyl)-3-(2-methyl-1-benzofuran-7-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(3S,4R)-4-(hydroxymethyl)-1-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]piperidin-3-ol
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}propanamide
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-phenylethan-1-one
4-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane