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N-methyl-2-(3-methyl-2-oxopyrrolidin-1-yl)-N-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}acetamide
N-(1-{7-[(4-methoxy-3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)-1-methylpiperidine-4-carboxamide
{[7-chloro-2-(2-methoxyphenyl)quinolin-3-yl]methyl}(1H-imidazol-2-ylmethyl)methylamine
1-cyclopropyl-5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-(1,3-dimethyl-1H-pyrazol-4-yl)-2-[2-(3-methoxyphenyl)pyrrolidin-1-yl]acetamide
N-{[5-(benzylsulfanyl)-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl]methyl}naphthalene-1-carboxamide
2-methyl-1-(1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazole
1-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
3-[(3-chlorophenyl)methyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
5-[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-4-yl]-5-ethyl-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2,2-dimethyl-N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propanamide
N-(2-{1-[(3-hydroxyphenyl)methyl]piperidin-3-yl}ethyl)pyridine-2-carboxamide
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(methylsulfanyl)acetamide
N-[3-(azepan-1-yl)propyl]-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
7-{[6-(hydroxymethyl)-1,4-oxazepan-4-yl]methyl}-2-methyl-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
1-[1-(2-chlorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-3-(4-methylpiperazin-1-yl)propan-1-one
4-[1-(4-chlorophenyl)cyclopropanecarbonyl]-7-(3,4-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
(2R,3R,6R)-3-(4-methylphenyl)-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
5-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-5-ethyl-3-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]imidazolidine-2,4-dione
2-{[(3-fluorophenyl)methyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
5-(2,6-dimethoxyphenyl)-N-(pyridin-4-ylmethyl)-1,2,4-triazin-3-amine
9-(2-chloro-5-fluorobenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-4-(thiophen-2-yl)butan-1-one
(1S,2S,3R,4R)-3-[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]bicyclo[2.2.1]heptan-2-amine
2,2-diphenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
N-(5-methyl-1,2-oxazol-3-yl)-2-[(2S,6S)-4-methyl-2,6-bis(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-oxoacetamide
{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
3-[(3,5-dimethylphenyl)methyl]-9-methoxy-N-[(2-methoxyphenyl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-1-{[4-(2-oxopyrrolidin-1-yl)phenyl]methyl}urea
2-(pyrrolidin-1-ylmethyl)-4-[(3,4,5-trimethoxyphenyl)methyl]-1,4-oxazepane
N-[2-(3-fluorophenyl)ethyl]-3-[(3S,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-(pyridin-4-ylmethyl)piperidin-3-yl]propanamide
5-({3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}methyl)-2-(methoxymethyl)pyrimidine
3-(1,2-oxazolidin-2-yl)-1-[3-(2-phenylethyl)piperidin-1-yl]propan-1-one
5-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]propan-1-one
2-[4-(2-cyclopropylpyrimidine-5-carbonyl)piperazin-1-yl]-1-(pyrrolidin-1-yl)ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
3-(5,6-dimethylpyrazin-2-yl)-2-methoxyquinoline
(1S,5R)-6-(5-methyl-1,3-oxazole-4-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
3-hydroxy-1-(2-phenylethyl)-3-{[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]methyl}piperidin-2-one
3-ethyl-1-[3-(4-fluorophenyl)phenyl]-3-[(3S,4R)-4-hydroxyoxolan-3-yl]urea
methyl[1-(4-methylpyridin-2-yl)propan-2-yl]{[6-(trifluoromethyl)pyridin-3-yl]methyl}amine
1-(cyclopropylmethyl)-N-[4-(3-methoxyphenyl)phenyl]piperidine-3-carboxamide
1-(2-methylpyridin-4-yl)-4-[(2-phenyl-1,3-oxazol-4-yl)methyl]-1,4-diazepane
4-{5-fluoro-2-[3-(pyridin-4-yl)azetidin-1-yl]pyrimidin-4-yl}morpholine
1-(6-{4-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperazin-1-yl}pyridin-3-yl)ethan-1-one
3-{[(2,2-difluoro-2H-1,3-benzodioxol-5-yl)methyl](ethyl)amino}-1λ6-thiolane-1,1-dione
6-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-triene-4-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
2-[3-(cyclopentylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(4-fluorophenyl)-2-oxoacetamide