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3-[1-(1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
1-{1-[(5-chlorothiophen-2-yl)sulfonyl]piperidin-3-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
5-(cyclopentylamino)-1-ethyl-N-(furan-2-ylmethyl)-N-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-methyl-N-[2-(morpholin-4-yl)ethyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
1-(cyclohex-3-ene-1-carbonyl)-4-(2-methylphenoxy)piperidine-4-carboxylic acid
4-{2-[4-(benzyloxy)-3-fluorophenyl]pyridine-4-carbonyl}morpholine
4-[3-(3-fluorophenoxymethyl)piperidine-1-carbonyl]-2-methoxypyridine
2-[ethyl({[(3R,4R)-4-(hydroxymethyl)-1-[2-(morpholin-4-yl)benzoyl]pyrrolidin-3-yl]methyl})amino]ethan-1-ol
2-(2-amino-6-methylpyrimidin-4-yl)-7-[(2,3-dimethoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-methyl-1,3-thiazole-5-carboxamide
1-(2-methoxy-6-methylbenzoyl)-3-(3-methoxypropyl)piperidine
2-{[(2-chlorophenyl)methyl]sulfanyl}-1-[2-(2-hydroxyethyl)piperidin-1-yl]ethan-1-one
4,6-dimethyl-2-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyridine-3-carbonitrile
(4aS,7aR)-1-(furan-3-carbonyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-(3,6-dimethylpyrazin-2-yl)-4-{spiro[2.3]hexane-1-carbonyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(1-methyl-1H-pyrazol-4-yl)-4-[2-(pyridin-3-ylmethyl)pyrrolidine-1-carbonyl]quinoline
4-bromo-N-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]benzamide
2-cyclobutanecarbonyl-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-tert-butyl-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carboxamide
N-methyl-N-[(5-propyl-1H-pyrazol-3-yl)methyl]-1,4-dithiepan-6-amine
4-(1-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)-1,2-dihydrophthalazin-1-one
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(2-oxoimidazolidin-1-yl)acetamide
N-[(5-ethylpyridin-2-yl)methyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(1R,5R)-6-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{2-[1-(pyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl]phenyl}ethan-1-one
1-{2-[3-(1H-pyrazol-3-yl)piperidine-1-carbonyl]phenyl}-1,3-diazinane-2,4-dione
5-[1-(5-acetylthiophene-3-carbonyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-methylimidazolidine-2,4-dione
1'-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
N-(2-chloro-4,6-dimethylphenyl)-3-[(4-methylpiperazin-1-yl)methyl]piperidine-1-carboxamide
2-amino-6-(2,5-dimethylthiophen-3-yl)-4-(1H-imidazol-4-yl)pyridine-3-carbonitrile
7-[(5-ethylfuran-2-yl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
5-[4-(1,4-diazepan-1-ylmethyl)phenyl]thiophene-2-sulfonamide
1-{2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-1,4-diazepan-5-one
1-(4-chloro-2-methylphenyl)-3-[(3S,5S,9R)-2,8-dioxo-1,7-diazatricyclo[7.3.0.03,7]dodecan-5-yl]urea
methyl[2-(phenylsulfanyl)ethyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
4-(benzyloxy)-1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
3-(1H-1,3-benzodiazol-2-ylmethyl)-N-(5-methyl-1,3,4-thiadiazol-2-yl)piperidine-1-carboxamide
2,3-dimethoxy-N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-[(2R,3R)-1'-(1,3-benzothiazol-2-ylmethyl)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
{[(3R,4S)-4-cyclopropyl-1-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]pyrrolidin-3-yl]sulfamoyl}dimethylamine
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-methylthiophen-2-yl)methyl]amine
3-[(2R,3R,6R)-5-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
1-{3-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
(2R,6R)-4-[2-(trimethyl-1H-pyrazol-1-yl)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
3-[(2R,6S)-2,6-dimethylmorpholin-4-yl]-1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}propan-1-one
(3S,4S)-4-propyl-1-(pyridine-3-sulfonyl)pyrrolidine-3-carboxylic acid
8-(5-acetylthiophene-2-carbonyl)-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-chloro-3-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidine-1-carbonyl}-1,2-dihydropyridin-2-one
N,N-dimethyl-3-(2-oxo-5,5-diphenylpiperidin-1-yl)propanamide
3-(2-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidin-1-yl}-2-oxoethyl)-1,3-oxazolidin-2-one