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3-(2-hydroxyphenyl)-N-[3-(1H-indol-1-yl)propyl]-1H-pyrazole-5-carboxamide
1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
N-ethyl-2-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}acetamide
5-fluoro-3,8-dimethyl-2-{4-[(2-methyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}quinoline
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]benzamide
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
4-ethyl-N,N-dimethyl-6-(4-{[(2-methyloxolan-2-yl)methyl]amino}piperidin-1-yl)pyrimidin-2-amine
1-benzyl-5-methanesulfonamido-2-methyl-N-(2-methylpropyl)-1H-1,3-benzodiazole-7-carboxamide
5-benzyl-2-methyl-4-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperidin-3-yl}pyrimidine
8-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-2-[(4-chlorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
7-{[4-(2-methanesulfonylethyl)piperazin-1-yl]methyl}-2,3-dimethyl-1H-indole
1-(2,2-diphenylethyl)-5-[2-(ethylamino)ethyl]pyrrolidin-2-one
5-(methanesulfonylmethyl)-2-(3-methyl-1H-pyrazol-5-yl)pyridine
3-(3-chlorophenyl)-N-(2-methoxyethyl)-3-phenylpropanamide
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)pyrazolo[1,5-a]pyridine-7-carboxamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
6-{4-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperazin-1-yl}pyrazine-2-carboxamide
2-(4-{[7-chloro-2-oxo-1-(prop-2-yn-1-yl)-1,2-dihydroquinolin-3-yl]methyl}piperazin-1-yl)-N-(propan-2-yl)acetamide
1-[5-(5-chlorothiophen-2-yl)-1H-1,2,4-triazol-1-yl]butan-2-ol
5-{7-methylimidazo[1,2-a]pyridin-2-yl}-3-(oxolan-2-ylmethyl)-1,2,4-oxadiazole
4-{2-[1-(3-fluorophenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}pyridine
8-[2-(3,5-dimethyl-1H-pyrazol-4-yl)acetyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-cyclopentyl-3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidine-1-carboxamide
(3R,9aR)-3-[(4-hydroxyphenyl)methyl]-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-{7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-5-phenylpentan-1-one
[(3R,4R)-1-(1-methyl-1H-1,3-benzodiazole-5-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
{5-[3-(hydroxymethyl)-3-propylpiperidine-1-carbonyl]-1H-1,3-benzodiazol-2-yl}methanol
1-ethyl-5-[4-(1H-indol-3-yl)butan-2-yl]-N-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
(1R,7S)-3-(2,2-dimethylpropyl)-N-methyl-N-(1,2-oxazol-5-ylmethyl)-4-oxo-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
1-(3-{[6-(piperidin-1-yl)pyrimidin-4-yl]amino}propyl)piperidin-3-ol
2-[1-({3-ethoxy-4-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-3-oxopiperazin-2-yl]-N-methylacetamide
N-ethyl-3-methyl-4-oxo-N-[2-(pyrrolidin-1-yl)ethyl]-3,4-dihydrophthalazine-1-carboxamide
(3S)-N,N-dimethyl-1-[(1-propyl-1H-imidazol-2-yl)methyl]azepan-3-amine
2-{5-[methoxy(phenyl)methyl]-3-(pyridin-4-yl)-1H-1,2,4-triazol-1-yl}acetic acid
6-cyclopropyl-N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}pyrimidin-4-amine
N-[3-(furan-2-yl)-3-phenylpropyl]-2-({6-[4-(pyridin-2-yl)piperazin-1-yl]pyridazin-3-yl}oxy)acetamide
2-(2-chloro-6-fluorophenyl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylacetamide
1-(2,3-dihydro-1H-inden-2-yl)-3-(2-methoxyethyl)-5-[3-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazole
2-[2-methyl-4-oxo-1-(oxolan-2-ylmethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]-N-(pyridin-2-ylmethyl)acetamide
5-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
N-{2-[1-(4-methyl-2-phenylpyrimidine-5-carbonyl)piperidin-2-yl]ethyl}acetamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1,2,2-trimethylpyrrolidin-3-yl)methyl]benzamide
2-({3-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)carbamoyl]phenyl}amino)acetic acid
3-{1-[(5-acetylthiophen-3-yl)methyl]piperidin-4-yl}-N-[(1-ethylpyrrolidin-2-yl)methyl]propanamide
(1R,5S)-6-{[3-(4-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-6-azabicyclo[3.2.1]octane
N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]-4-[(2-methylprop-2-en-1-yl)oxy]benzamide
1-[(1S,5R)-6-{4-[(dimethylamino)methyl]benzoyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
[(1-{[1-(thiophen-3-ylmethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]urea
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl){[2-(propan-2-yl)pyrimidin-5-yl]methyl}amine