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N-{1-[7-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}-2-methylfuran-3-carboxamide
2-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]-8-methyl-2,8-diazaspiro[5.5]undecane
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][(1R)-1-(3-methoxyphenyl)ethyl]amine
2-[2-chloro-4-({3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)phenoxy]acetamide
{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-N,5-dimethyl-N-(1,2-oxazol-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
8-[(3Z)-hex-3-en-1-yl]-2H,5H,6H,7H,8H-[1,3]dioxolo[4,5-g]quinolin-6-one
N-[(4-fluorophenyl)methyl]-N-(3-methoxypropyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
3-[(1R,2S)-2-(methoxymethyl)cyclopentyl]-1-(naphthalen-1-yl)urea
2-(1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-1,3-benzoxazole
2-benzyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,3-benzoxazole-5-carboxamide
N-({5-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-methyl-3-({3-[2-(methylsulfanyl)ethyl]-1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl}methyl)imidazolidine-2,4-dione
1-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidin-1-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
2-benzyl-9-(oxane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(oxan-2-ylmethyl)-1H-pyrazole-3-carboxamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
7-(morpholin-4-ylmethyl)-4-[(2-phenyl-1,3-thiazol-5-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
[(3R,4S)-4-[(4-ethylpiperazin-1-yl)methyl]-1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-3-yl]methanol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[1-(pyridin-4-yl)propyl]amine
3-[(4-fluorophenyl)methyl]-1-(quinoxalin-2-yl)piperidine-3-carboxylic acid
2-{4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
5-(oxolan-2-yl)-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]thiophene-2-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
2-(4-fluorophenyl)-N-{2-[7-(3-phenylpropyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}acetamide
N,N-dimethyl-1-{4-[1-(3-methylphenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}pyrrolidin-3-amine
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-3-[4-(methylsulfanyl)benzoyl]piperidine
N-[2-methoxy-4-(1H-pyrazol-3-yl)phenyl]acetamide
(4aS,8aS)-2-[(2-propoxynaphthalen-1-yl)methyl]-decahydro-2,7-naphthyridin-4a-ol
1-(2-fluorophenyl)-4-(piperidin-3-yl)piperazine
1-{4-[(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperazin-1-yl}ethan-1-one
1-(4-{[methyl(pyrazin-2-ylmethyl)amino]methyl}phenoxy)-3-(piperidin-1-yl)propan-2-ol
1-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
2-{4-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]piperidin-1-yl}-6-fluoro-4-methylquinazoline
N-(5-tert-butyl-2-methoxyphenyl)-4-(2-methoxyacetyl)-1,4-diazepane-1-carboxamide
5-{3-benzyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl}-3-ethyl-4-methyl-1H-pyrazole
N-benzyl-N-(cyclopropylmethyl)-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)piperidine-3-carboxamide
1-(5-ethyl-1,2-oxazole-3-carbonyl)-3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine
4-[3-(1H-pyrazol-1-yl)propyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-[5-(2,5-difluorophenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]pyridine
{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}(pyridin-2-ylmethyl)amine
N-methyl-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}-2-(pyrrolidin-3-yl)benzamide
2-{1-[(2-ethoxyphenyl)methyl]-4-(1H-indol-2-ylmethyl)piperazin-2-yl}ethan-1-ol
3-(2-chlorophenyl)-3-[2-(4-cyclopentyl-3-oxopiperazin-1-yl)-2-oxoethyl]-1-[2-(dimethylamino)ethyl]pyrrolidine-2,5-dione
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(2-oxo-2-{2-[2-(thiophen-2-yl)ethyl]piperidin-1-yl}ethyl)imidazolidine-2,4-dione
2-(5-{2-[2-(1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
methyl 1-(2-methoxyethyl)-3-(3-phenylpropanamido)-5-[(2-phenylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[2-(2-cyclopentylacetamido)ethyl]-N-(2-methylphenyl)-1H-1,2,3-triazole-4-carboxamide
2-methyl-5-({3-[2-(pyridin-2-yl)piperidine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)-1,3-benzothiazole