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2-{[3-(2-methylphenyl)phenyl]methyl}-octahydropyrrolo[1,2-a]piperazine
(2S)-1-{1-[(2E)-3-phenylprop-2-en-1-yl]-1H-1,2,3-triazole-4-carbonyl}pyrrolidine-2-carboxamide
2-(2-oxoazepan-1-yl)-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)acetamide
5-methoxy-2-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-4H-pyran-4-one
2-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methoxyphenol
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[(2-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
4-{1-[4-(1H-pyrazol-3-yl)benzoyl]azetidin-3-yl}pyridine
5-(2,5-dimethylphenoxymethyl)-N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-1,2-oxazole-3-carboxamide
(4aR,7aS)-1-benzyl-4-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(4-methoxyphenyl)methyl]-1-methyl-8-(quinolin-7-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2R,6R)-11-methoxy-4-[3-(1H-pyrazol-1-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(prop-2-en-1-yl)-3-[3-(propan-2-yloxy)benzoyl]piperidine-1-carboxamide
2-(dimethylamino)-8-[(4-phenylphenyl)methyl]-1,3,8-triazaspiro[4.5]dec-1-en-4-one
N5-(butan-2-yl)-1-cyclopentyl-N3-methyl-4-oxo-N3-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-[2-methyl-6-(2-methylpropyl)pyrimidine-4-carbonyl]piperidin-3-amine
1-[(4-ethynylphenyl)methyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
3-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1H-pyrazol-5-amine
(2S,4R)-1-[2-(adamantan-1-ylsulfanyl)acetyl]-4-amino-N-methylpyrrolidine-2-carboxamide
N-methyl-2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-(1,2-oxazol-5-ylmethyl)acetamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-methoxy-N-[2-(methylsulfanyl)ethyl]benzamide
(1S,5R)-6-[(3-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}benzoic acid
N-(1,3-benzothiazol-2-yl)-3-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}propanamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-4-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperazine-1-carboxamide
3-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-1-methyl-1,2-dihydroquinolin-2-one
1-[(3-chloro-2,4-difluorophenyl)methyl]-4-methylpiperidine-4-carbonitrile
8-(1-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-imidazol-2-yl)quinoline
1-cyclopentyl-4-[3-(pyridin-3-yl)azetidine-1-carbonyl]pyrrolidin-2-one
8-(4-aminopyridine-2-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{2-[4-(2-phenyl-1,3-oxazol-4-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1,2-dihydrophthalazin-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(3-fluorophenyl)-N-(pyridin-3-ylmethyl)-1,3-benzoxazole-5-carboxamide
6-(2-chlorophenyl)-N,7-dimethyl-N-(2-methylpropyl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-amino-6-(5-methyl-1H-1,3-benzodiazol-2-yl)-4-(oxolan-3-yl)pyridine-3-carbonitrile
(4aS,7aR)-1-(5-fluoro-2-methylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(azepan-1-yl)ethyl]-N-methyl-2-(trifluoromethyl)pyrimidin-4-amine
(4aS,8aR)-1-[3-(methylsulfanyl)propyl]-6-(1,3-thiazol-2-yl)-decahydro-1,6-naphthyridin-2-one
3-(2-methylpropyl)-4-[5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carbonyl]morpholine
4-(2-{3,9-diazaspiro[5.5]undecan-3-yl}-2-oxoethyl)morpholin-2-one
1-[7-(1-benzothiophen-3-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-methyl-2-(methylamino)propan-1-one
1-[3-(4-{[(1R,2S)-2-(methoxymethyl)cyclopentyl]amino}piperidin-1-yl)phenyl]pyrrolidin-2-one
N4-cyclopropyl-6-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]pyrimidine-2,4-diamine
5-methanesulfonyl-N-(1-methanesulfonylpiperidin-4-yl)-2-methylpyrimidin-4-amine
2-(2-hydroxyphenoxy)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)ethan-1-one
methyl (2S)-2-({1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazol-4-yl}formamido)-2-phenylacetate
2-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}-3-methoxyphenol
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-(1-{6-phenylimidazo[2,1-b][1,3]thiazole-3-carbonyl}piperidin-3-yl)-1H-1,3-benzodiazole
3-phenyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
N-[(1R,3R)-3-aminocyclopentyl]-1-[2-(dimethylamino)ethyl]-3-methyl-1H-pyrazole-5-carboxamide