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5-(2-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-2-oxoethyl)pyrrolidin-2-one
1-methyl-6-propyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}[3-(2-methyl-1H-imidazol-1-yl)-1-phenylpropyl]amine
(2,2-dimethylpropyl)[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
[(5-{1-[1-(difluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]dimethylamine
N-{[7-(5-acetylthiophen-2-yl)-5-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(3-methoxyphenyl)propanamide
1-{4-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-1,4-diazepan-1-yl}ethan-1-one
1-[2-(3-fluorophenyl)ethyl]-N-[2-(2-methylphenyl)ethyl]-6-oxopiperidine-3-carboxamide
5-ethyl-N4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-6-methylpyrimidine-2,4-diamine
6-(azepan-1-yl)-N-[2-(morpholin-4-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
3-cyclopropyl-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-1H-pyrazole-5-carboxamide
5-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}-2-(pyrrolidin-1-yl)pyrimidine
N-methyl-2-(morpholin-3-yl)-N-(1,2-oxazol-5-ylmethyl)acetamide
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
3-(2,3-dihydro-1,4-benzodioxin-6-ylsulfanyl)-N-methyl-N-[2-(oxan-4-yl)ethyl]propanamide
N-[2-(dimethylamino)ethyl]-N-[(3-methylthiophen-2-yl)methyl]-4-oxo-1,4-dihydroquinoline-2-carboxamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,6-dichlorobenzamide
(2S)-2-({[4-(carbamoylmethoxy)phenyl]methyl}amino)propanamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(piperidin-1-yl)-2,3-dihydro-1H-indene-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)acetamide
7-[2-(aminomethyl)-7-chloro-2,3-dihydro-1-benzofuran-5-yl]-3,4-dihydro-2H-1-benzopyran-4-one
1-[(2,6-difluoro-3-methoxyphenyl)methyl]-3-(1-methyl-1H-1,2,4-triazol-3-yl)urea
ethyl 1-[6-(1-benzothiophen-2-yl)-2-(morpholin-4-yl)pyridine-3-carbonyl]piperidine-3-carboxylate
2-(dimethyl-1,3-thiazol-5-yl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-methylbutanamide
3-(4-methylphenyl)-1-[7-(2-methylphenyl)-9-(oxolan-3-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
N-({3-methoxy-4-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)-1,3-dimethyl-N-(pyridin-2-ylmethyl)-1H-pyrazole-5-carboxamide
1-(4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-4-phenylpiperidine-4-carbonitrile
1-(4-benzylpiperidin-1-yl)-3-[1-(5-methoxyfuran-2-carbonyl)piperidin-4-yl]propan-1-one
5-{4-[2-(5-tert-butyl-1H-pyrazol-3-yl)-1H-imidazol-1-yl]phenoxy}-1H-1,2,3,4-tetrazole
3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-[3-(pyridin-3-yloxy)propyl]propanamide
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-(3-hydroxyphenyl)ethan-1-one
N-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)-5-(pyrimidin-5-yl)pyrimidin-2-amine
N-cyclopropyl-N-propyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-{[(6-chloropyridin-3-yl)carbamoyl]amino}-N,N,3-trimethylbutanamide
N-[2-(5-chloro-4-methyl-1,3-thiazol-2-yl)ethyl]-1-methyl-1H-indole-6-carboxamide
N-[2-(dimethylamino)-5,6,7,8-tetrahydroquinazolin-5-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
4-acetyl-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)benzamide
4-(4-chlorophenoxy)-N-[(2R)-oxolan-2-ylmethyl]piperidine-4-carboxamide
1-({1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(piperidin-1-yl)propan-2-ol
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
8-{5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
1-{[3-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
3-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
3-[3-({[1-(thiophen-2-yl)propan-2-yl]amino}methyl)-1H-indol-1-yl]propanamide
N-({1-[3-(1,2-oxazinan-2-yl)propanoyl]piperidin-3-yl}methyl)thiophene-2-sulfonamide
2-(3-chlorophenyl)-N-{[5-(3,6-dimethylpyrazin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
{1-ethyl-5-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
3-methyl-1-[(4-methylphenyl)methyl]-4-[3-(pyridin-3-yl)propanoyl]piperazin-2-one