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1-methyl-5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-pyrrole-3-carbonitrile
2-[(2-ethyl-4-methyl-1,3-oxazol-5-yl)formamido]-N-(4-fluoro-2-methylphenyl)propanamide
1-[(3-fluorophenyl)methyl]-6-oxo-N-[3-(pyridin-2-yl)propyl]piperidine-3-carboxamide
2-[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
N-{1-[(4-chlorophenyl)methyl]-4-methyl-1H-pyrazol-5-yl}-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
4-(5-methylthiophene-2-carbonyl)-2-(piperidin-1-ylmethyl)-1,4-oxazepane
N-[1-(1-benzylpiperidin-4-yl)-1H-pyrazol-5-yl]-4-phenylbutanamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-(2-hydroxyethyl)-N-(5-methyl-2,1,3-benzothiadiazol-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
5-(azepane-1-carbonyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-2-one
(3R,4R)-1-{[6-(dimethylamino)pyridin-3-yl]methyl}-3-methyl-4-(oxan-4-yl)piperidin-4-ol
1-acetyl-N-[(3R,4S)-4-cyclopropyl-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]piperidine-4-carboxamide
N-ethyl-1-(3-methylbenzenesulfonyl)-N-(pyridin-4-ylmethyl)piperidin-3-amine
2-(4-chlorophenoxymethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-[(2R,3R)-1'-[(2-hydroxynaphthalen-1-yl)methyl]-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]thiophene-3-carboxamide
1-(7-methanesulfonyl-4-methylquinazolin-2-yl)-N-[2-(methylsulfanyl)ethyl]piperidine-3-carboxamide
(3R,4S)-4-cyclopropyl-N,N-dimethyl-1-(oxan-4-yl)pyrrolidin-3-amine
N-(2,3-dihydro-1H-inden-2-yl)-2,6-dimethoxy-N-methylpyrimidine-4-carboxamide
4-(azocan-1-yl)-5-methyl-N-[2-(methylsulfanyl)ethyl]thieno[2,3-d]pyrimidine-6-carboxamide
(4aR,7aS)-1-(2-methylpropanoyl)-4-[2-(6-methylpyridin-2-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-1-methyl-3-(2-methylpropyl)-N-(3-phenylprop-2-yn-1-yl)-1H-pyrazole-5-carboxamide
N,3-dimethyl-1-propyl-N-(thian-4-yl)-1H-pyrazole-4-carboxamide
(3S,4R)-4-(pyridin-4-yl)-1-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]pyrrolidine-3-carboxylic acid
1-[3-(3-fluoropyridin-2-yl)phenyl]ethan-1-one
(2S,4R)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-methylthiophen-2-yl)methyl]amino}pyrrolidine-2-carboxamide
{[2-(benzylsulfanyl)pyrimidin-5-yl]methyl}[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]methylamine
(1S,5R)-6-[(2-ethyl-1,3-thiazol-4-yl)methyl]-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
{[2-cyclohexylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)[2-(morpholin-4-yl)ethyl]amine
4-(1-benzylpyrrolidin-3-yl)-1-(3-methoxyphenyl)-6-methylpiperazin-2-one
2-(4-methyl-6-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}pyrimidin-2-yl)phenol
5-(3-methylbutyl)-5-[1-(3-phenoxypropanoyl)piperidin-4-yl]-3-(pyridin-2-ylmethyl)imidazolidine-2,4-dione
2-{5-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl}ethan-1-ol
2-{1-[(4-methylphenyl)methyl]-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-3-yl}acetamide
5-(4-{3H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}phenyl)-8-methoxy-2-methylquinoline
N-(1-methyl-1H-pyrazol-4-yl)-4-({methyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)benzamide
4-hydroxy-N-[(4-phenyloxan-4-yl)methyl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
3-(1H-1,2,3-benzotriazol-1-yl)-1-[4-(2,6-dimethylpyridin-4-yl)piperazin-1-yl]propan-1-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(methylsulfamoyl)benzamide
N-{[2-(3-chlorophenyl)-7-methylquinolin-3-yl]methyl}-N-(3-methoxypropyl)propanamide
2-(3-fluorophenyl)-N-[(7-{[3-(2-hydroxyethoxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]acetamide
3-methyl-1-[3-(phenylamino)piperidin-1-yl]but-2-en-1-one
1-methyl-N-{[5-methyl-2-(2-phenylmethanesulfonamidophenyl)-1,3-oxazol-4-yl]methyl}-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-[(2-ethoxyphenyl)methyl]-4-(pyridin-3-yl)pyrimidin-2-amine
(3S,4R)-3-ethyl-4-methyl-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]piperidin-4-ol
methyl (3S)-3-amino-4-[4-(dimethylamino)-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-4-oxobutanoate
(3S)-N-tert-butyl-2-{2-[(dimethylcarbamoyl)amino]acetyl}-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
3-(3-acetylphenyl)-1-methyl-6-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{4-[(4-chlorophenyl)methyl]piperazin-1-yl}-3-(pyridin-4-yl)propan-1-one
8-[(4-methoxypyridin-2-yl)methyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-(2-chlorophenyl)-1-[2-(dimethylamino)ethyl]-3-[2-oxo-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]pyrrolidine-2,5-dione