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2-{1-methyl-5-[4-(morpholin-4-yl)piperidin-1-yl]-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl}-1,2,3,4-tetrahydroisoquinoline
1-(5-chloropyridin-2-yl)-4-[4-(pyrrolidine-1-carbonyl)pyridin-2-yl]piperazine
4-{2-oxo-2-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethyl}piperazin-2-one
2-[6-(cyclopentylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzoic acid
{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}(methyl)[(5-propyl-1H-pyrazol-3-yl)methyl]amine
1-(2,2-dimethylpropyl)-4-[(2-methylphenyl)methyl]-1,4-diazepan-5-one
2-(methylamino)-N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]pyrimidine-5-carboxamide
N-(1-{1-[(1-methyl-1H-indol-3-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
(3S)-1-(1-benzothiophene-5-carbonyl)-N,N-dimethylazepan-3-amine
4-[(1E)-3,3-dimethylbut-1-en-1-yl]-N,N-dimethylbenzamide
methyl 6-({methyl[1-(4-methylpyridin-2-yl)propan-2-yl]amino}methyl)pyridine-2-carboxylate
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-3,4-dimethyl-5-sulfamoylbenzamide
1-{1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}-1,4-diazepane
2-(3-fluoro-4-methoxyphenyl)-2-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]acetic acid
methyl 4-{4-[4-(methylsulfanyl)benzoyl]piperazin-1-yl}benzoate
N-[(3-chlorophenyl)methyl]-1-(2-methoxyethyl)-N-methylpyrrolidine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-5-[(oxan-2-ylmethoxy)methyl]-1H-1,2,4-triazole
5-methoxy-2-{[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4H-pyran-4-one
N,2-dimethyl-2-[(2-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,3-oxazol-4-yl)formamido]propanamide
N-(2-methoxyethyl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
4-{4-[4-(2-hydroxyethyl)piperazin-1-yl]piperidin-1-yl}-N-(1-phenylethyl)benzamide
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methyl-N-(2-methylpropyl)thiophene-2-carboxamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(6-methoxy-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-1-methylurea
N,3-dimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
methyl 5-{[(4-acetamidophenyl)methyl]amino}-3-(2-methoxyacetamido)-1-(3-phenylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
13-(3-chloro-4-propoxyphenyl)-5-thia-2,7,10-triazatricyclo[6.5.0.02,6]trideca-1(8),3,6-trien-11-one
N-methyl-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
1-[1'-(5-fluoropyridine-3-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
N-ethyl-N-[(3S,4R)-4-hydroxyoxolan-3-yl]-3-(1,2-oxazinan-2-yl)propanamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-{[5-(propan-2-yl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxylate
1-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]-3-phenoxypropan-1-one
{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
3-{2-[2-(ethylsulfanyl)pyrimidin-5-yl]-1H-imidazol-1-yl}-4-hydroxybenzonitrile
6-(3-methoxy-2-methylbenzoyl)-2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
2-[N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamido]-2-(pyridin-3-yl)acetic acid
1-cyclohexyl-4-[6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonyl]-1,4-diazepane
1-{5-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]thiophen-2-yl}ethan-1-one
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(diethylamino)ethyl]-N-methyl-1H-pyrazole-3-carboxamide
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(2-methoxyethyl)-2-methyl-1-benzofuran-7-carboxamide
[(1-cyclopentylpiperidin-4-yl)methyl][(3-ethoxy-4-methoxyphenyl)methyl](oxolan-2-ylmethyl)amine
1-ethyl-8-[(3-hydroxyphenyl)methyl]-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[(2,4-difluorophenyl)methyl]-N-[2-(3-methoxyphenyl)phenyl]piperidine-4-carboxamide
3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)-N-[3-(4-methyl-1,3-thiazol-5-yl)propyl]propanamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-(furan-3-ylmethyl)-N-methylbenzamide
2-(1H-indol-3-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]ethan-1-one
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-ethyl-N-methylpyridin-2-amine
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-4-phenylbenzamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2-[ethyl(methyl)amino]propan-1-one
methyl (2S,4S)-1-(naphthalen-1-ylmethyl)-4-propanamidopyrrolidine-2-carboxylate
4-(cyclopropylmethyl)-1-[2-(dimethyl-1,2-oxazol-4-yl)ethyl]-3-(propan-2-yl)-1,4-diazepan-5-one