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2-cyclopropyl-N-[2-(1H-imidazol-1-yl)ethyl]-N-methyl-1,3-benzoxazole-6-carboxamide
3-[2-(4-benzylpiperazin-1-yl)-2-oxoethyl]-1-[2-(dimethylamino)ethyl]-3-(3-fluorophenyl)pyrrolidine-2,5-dione
1-{[3-({1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}oxy)phenyl]methyl}-4-(pyridin-3-ylmethyl)piperazine
1-[3-(3-methoxyphenyl)phenyl]-N-(1,3-thiazol-2-ylmethyl)piperidin-4-amine
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(pyridin-4-yl)propanamide
2-{[2-(trifluoromethyl)phenyl]methyl}-9-oxa-2-azaspiro[5.5]undecane
7-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-(2,5-dioxoimidazolidin-4-yl)-N-[(4-methoxyphenyl)methyl]-N-propylacetamide
3-hydroxy-N-[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]pyridine-2-carboxamide
3-[(3R,4S)-1-[(3-chloro-4-methoxyphenyl)carbamoyl]-4-(dimethylamino)piperidin-3-yl]propanoic acid
1-[4-(3-methoxybenzoyl)piperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-chloro-4-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}-N-[2-(pyrazin-2-yl)ethyl]benzamide
3-(furan-2-yl)-3-phenyl-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}propanamide
4-{3-[(2,3-dimethylquinoxalin-6-yl)formamido]propyl}-1,2,5-oxadiazole-3-carboxylic acid
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-(1-methyl-1H-pyrrole-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[(2-hydroxyethyl)sulfanyl]-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-2-ethylpyrimidine
(3R,4R)-4-cyclobutyl-3-methyl-1-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}piperidin-4-ol
4-[(3,5-difluorophenyl)methyl]-7-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
4-[2-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-2-phenylethyl]phenol
3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-(propan-2-yl)propanamide
4-(difluoromethoxy)-N-(isoquinolin-5-ylmethyl)-N-methylbenzamide
3-{[4-(3-chlorophenyl)-5-({methyl[(6-methylpyridin-2-yl)methyl]amino}methyl)-4H-1,2,4-triazol-3-yl]sulfanyl}propan-1-ol
5-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2-(pyridin-4-yl)pyrimidine
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-indole-5-carboxamide
4-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]pyrimidin-2-amine
5-methyl-1'-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(1H-imidazol-2-ylmethyl)-2-(1-oxo-4-phenyl-1,2-dihydrophthalazin-2-yl)acetamide
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methylpyridine-3-carbonyl)pyrrolidin-3-yl]methanol
N-{[7-chloro-2-(4-methoxyphenyl)quinolin-3-yl]methyl}-2-(2,5-dimethoxyphenyl)-N-(oxolan-2-ylmethyl)acetamide
2-methyl-5-[2-(3,4,5-trimethoxyphenyl)-1H-imidazol-1-yl]pyridine
2-(3,3-dimethylbutanoyl)-7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
2-[2-(1H-imidazol-1-yl)ethyl]-1-[1-(4-methylphenyl)cyclopropanecarbonyl]piperidine
2-[2-oxo-4-(4-oxo-3,4-dihydrophthalazine-1-carbonyl)piperazin-1-yl]benzonitrile
1-methyl-2-(morpholin-4-yl)-5-[3-(pyridin-2-yl)azetidine-1-carbonyl]-1H-1,3-benzodiazole
N-(2-{1-[(1-methyl-1H-pyrazol-4-yl)sulfonyl]piperidin-2-yl}ethyl)acetamide
1-(2-methoxyethyl)-8-(2-methylpropyl)-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]methyl}-1H-pyrazole-3-carboxylic acid
5-chloro-1,3-dimethyl-4-{[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-pyrazole
5-{1-cyclohexyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-4-methyl-1,3-oxazole
1-[2-(dimethylamino)ethyl]-5-oxo-N-[1-(pyridin-4-ylmethyl)piperidin-4-yl]pyrrolidine-3-carboxamide
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)-2-(methylamino)acetamide
(1H-indol-5-ylmethyl)(methyl)[(1-phenyl-1H-pyrazol-4-yl)methyl]amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-(propan-2-yl)piperidine-4-carboxamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)acetamide
2-amino-6-(3,4-difluorophenyl)-4-[2-(ethylamino)pyrimidin-5-yl]pyridine-3-carbonitrile
2-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-4-(piperidine-1-carbonyl)pyridine
N-[(2R,3R)-1'-(1-phenylcyclopropanecarbonyl)-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
N-methyl-6-(6-methylpyridazin-3-yl)-4-(pyrrolidine-1-carbonyl)-5H,6H,7H,8H-pyrido[4,3-d]pyrimidin-2-amine
1-[2-(4-chlorophenyl)morpholin-4-yl]-3-ethoxypropan-1-one