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2-(4-fluorophenyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
1-(2-fluorophenyl)-4-{1-[(3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl}piperazine
4-{2-[(4-methoxyphenyl)methyl]-1,3-benzoxazole-6-carbonyl}-1,4-diazepane-1-carbaldehyde
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-N-(1,1-dioxo-1λ6-thiolan-3-yl)piperidine-1-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-ethoxyethyl)pyrrolidin-3-yl]-1,1-dioxo-1λ6-thiane-4-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-{[5-(1-methanesulfonylpiperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}-4-methylpiperazine
1-(4,7-dimethylquinazolin-2-yl)-N-(2,2,2-trifluoroethyl)piperidine-3-carboxamide
1-{4-[(oxan-4-ylmethyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
7-[(2,3-difluorophenyl)methyl]-2-(4-methylpentanoyl)-2,7-diazaspiro[4.5]decan-6-one
2-(1-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)pyridine
2-[4-(2,5-dihydro-1H-pyrrol-1-yl)-2-(ethoxymethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetic acid
(1R,3S)-3-methoxy-7-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-7-azaspiro[3.5]nonan-1-ol
1-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(3R,4S)-1-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
(2S)-N-({2-[4-(2-methoxyphenyl)piperazin-1-yl]pyridin-3-yl}methyl)pyrrolidine-2-carboxamide
[(3R,4R)-1-(2-cyclopropylpyrimidine-5-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(3R,4S)-4-cyclopropyl-1-(4-ethyl-2-methyl-1,3-thiazole-5-carbonyl)-N,N-dimethylpyrrolidin-3-amine
N-cyclopropyl-3-(4-methyl-4H-1,2,4-triazol-3-yl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]propanamide
1-(1,4-dithiepan-6-yl)-3-[3-(trifluoromethyl)benzoyl]piperidine
5-[1-(2,3-dimethoxybenzoyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(3-methylbutyl)imidazolidine-2,4-dione
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-2,3-dimethoxybenzamide
1-[(2-phenyl-1,3-oxazol-4-yl)methyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-(1H-1,3-benzodiazol-2-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]propanamide
3-[methyl(1-methylpyrrolidin-3-yl)amino]-1-[4-(2-phenylethyl)piperidin-1-yl]propan-1-one
(3S,4R)-4-methyl-1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidine-3,4-diol
2-{1-[(4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(1H-imidazol-1-yl)propyl]acetamide
4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}butanamide
N-[(2R,3R)-2-methoxy-1'-[(4-methoxy-2,5-dimethylphenyl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]furan-2-carboxamide
3-(2-ethyl-5-oxopyrrolidin-2-yl)-N-[(3-phenyl-1H-pyrazol-4-yl)methyl]propanamide
(2R,3R,6R)-3-(4-methoxyphenyl)-N-(propan-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-{1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl}propanamide
N-[2-(4-methoxyphenyl)phenyl]-1-(pent-4-enoyl)pyrrolidine-2-carboxamide
(2S,4S)-4-amino-N-[(5-chloro-1-benzothiophen-3-yl)methyl]-1-methylpyrrolidine-2-carboxamide
N-[(1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methyl]acetamide
7-methyl-3-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-3,7,11-triazaspiro[5.6]dodecan-12-one
N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
1-[(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)methyl]pyrrolidin-2-one
4-[(3-methylphenyl)sulfanyl]-1-(3,3,3-trifluoropropyl)piperidine
2-(1-cyclopentyl-4-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-2-yl)ethan-1-ol
N-(furan-2-ylmethyl)-5,6-dimethyl-N-[2-(morpholin-4-yl)ethyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
2-methoxy-1-{4-[3-(pyridin-2-yl)azetidine-1-carbonyl]piperidin-1-yl}ethan-1-one
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}bis(pyridin-3-ylmethyl)amine
4-({1-[(3-acetylphenyl)methyl]piperidin-4-yl}oxy)-3-chloro-N-(2-methoxyethyl)benzamide
9-hydroxy-3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}-4H-pyrido[1,2-a]pyrimidin-4-one
(3S,4R)-1-(5-ethylthiophene-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-[(4,6-dimethylpyridin-3-yl)methyl]-2-methyl-6-(piperidin-3-yl)pyrimidin-4-amine
3-[2-(dimethylsulfamoyl)ethyl]-1-{3-[(trifluoromethyl)sulfanyl]phenyl}urea
N-cyclopropyl-N-{[4-methoxy-3-(pyridin-4-ylmethoxy)phenyl]methyl}-3-methylthiophene-2-carboxamide