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1-(cyclopropylmethyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)-2-(propan-2-yl)-1,4-diazepane
6-fluoro-2-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}quinolin-4-ol
[2-(diethylamino)ethyl](methyl)({3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)amine
N4,N4,5-trimethyl-N2-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidine-2,4-diamine
{1-[(6-chloro-2H-chromen-3-yl)methyl]-3-[(3-methoxyphenyl)methyl]piperidin-3-yl}methanol
(5S,9aS,9bS)-5-[4-(furan-2-yl)phenyl]-2-[(4-methoxyphenyl)methyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-5-oxo-1-(pyridin-2-ylmethyl)pyrrolidine-3-carboxamide
1-{[1-benzyl-2-(2-methylpropanesulfonyl)-1H-imidazol-5-yl]methyl}-4-(cyclopropylmethyl)piperazine
8-[6-(propan-2-yl)pyridin-2-yl]-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(3-methoxypropyl)-6-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-{[6-chloro-4-(pyrrolidin-1-yl)quinazolin-2-yl]methyl}-3-(furan-2-yl)-3-phenylpropanamide
N-[2-methyl-6-(propan-2-yl)phenyl]-2-[3-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
7-(2-methoxyethyl)-2-{[3-(methylsulfanyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1-oxa-8-azaspiro[4.6]undecane
6-methyl-4-{2-methyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}-1,2-dihydropyridin-2-one
2-(2,5-dimethoxyphenyl)-1,3-benzoxazole
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[1-(pyridine-3-carbonyl)piperidin-4-yl]-1,4-diazepane
5-(2,6-dimethylpyrimidine-4-carbonyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-methoxy-N-{2-[7-(quinolin-5-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}benzamide
6-(3-fluoro-4-methoxybenzoyl)-N-[(4-phenyloxan-4-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
3-[2-(4-fluorophenyl)morpholine-4-carbonyl]-6-(propan-2-yl)-1,2-dihydropyridin-2-one
4-(4-chlorophenoxy)-N-[(3S,4R)-4-methoxyoxolan-3-yl]piperidine-4-carboxamide
2-methoxy-N-[1-methyl-4-(2-oxo-1,3-oxazolidin-3-yl)-1H-indazol-3-yl]pyridine-4-carboxamide
2-[ethyl({[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl})amino]ethan-1-ol
1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-4-methyl-1,4-diazepan-5-one
1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-8-(pyridin-2-yl)-1,8-diazaspiro[4.5]decane
3-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-phenyl-1H-pyrazol-5-amine
5,7-dimethoxy-4-(4-methyl-1H-imidazol-5-yl)-1,2,3,4-tetrahydroquinolin-2-one
N-(2-hydroxy-2-phenylethyl)-N-methylspiro[2.3]hexane-1-carboxamide
1-(furan-2-ylmethyl)-N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}piperidine-4-carboxamide
8-(dimethyl-1,3-oxazole-5-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
2-(1-methyl-1H-imidazol-2-yl)-1-[(3-{[3-(trifluoromethyl)phenyl]methyl}-1,2,4-oxadiazol-5-yl)methyl]piperidine
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-phenoxyacetamide
N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-3-methylbut-2-enamide
N-cyclopropyl-N-[(3-ethoxyphenyl)methyl]-1-ethyl-1H-pyrazole-3-carboxamide
1-{1-[4-(pyridin-2-yl)piperazine-1-carbonyl]-6-azaspiro[2.5]octan-6-yl}-2-[3-(trifluoromethyl)phenyl]ethan-1-one
5-{2-[(prop-2-en-1-yl)amino]ethyl}-1-[2-(thiophen-2-yl)ethyl]pyrrolidin-2-one
N-[(3R,4R)-1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-hydroxypiperidin-4-yl]pyridine-4-carboxamide
3-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]-1-{2,7-dimethylimidazo[1,2-a]pyridine-3-carbonyl}piperidine
2-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-4-methylphenol
1-[(4-cyano-5-methyl-1H-pyrrol-2-yl)methyl]-4-(naphthalen-2-yloxy)piperidine-4-carboxylic acid
2-(2-methyl-1,3-thiazol-4-yl)-N-{[3-(3-methylbutyl)-3H-imidazo[4,5-b]pyridin-2-yl]methyl}acetamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[4-(1H-pyrazol-1-yl)butan-2-yl]amine
N-methyl-4-(pyridin-2-yl)-N-{[2-(pyrrolidin-1-ylmethyl)phenyl]methyl}pyrimidin-2-amine
1-benzyl-8-{[5-(hydroxymethyl)furan-2-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
({4-[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)piperidin-2-yl]phenyl}methyl)dimethylamine
N-[(2-fluorophenyl)methyl]-4-(4-{[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl)benzamide
({5-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]furan-2-yl}methyl)dimethylamine
5-phenyl-N-[(3,4,5-trifluorophenyl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
4-[(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-2-yl)methyl]morpholine