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4-(2,3,4,9-tetrahydro-1H-carbazole-7-carbonyl)-1,4-oxazepan-6-ol
2-methoxy-N-({5-methyl-2-[4-(2-phenylacetamido)phenyl]-1,3-oxazol-4-yl}methyl)-2-phenylacetamide
2-[4-(4-cyclopentylphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]acetamide
[2-(diethylamino)ethyl](ethyl)({1-[(2-fluorophenyl)methyl]-2-(propane-2-sulfonyl)-1H-imidazol-5-yl}methyl)amine
1-[5-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-2-methylphenyl]imidazolidin-2-one
3-{[1-(4-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1λ6-thiolane-1,1-dione
3-methyl-2-[3-(oxolan-3-yl)-1-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]-1H-indole
3-{1-[1-(3-aminopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-1-(2-chlorophenyl)urea
4-(4-methylpiperazin-1-yl)-6-(pyrimidin-5-yl)pyrimidin-2-amine
N-({3-methyl-7-[(2E)-3-phenylprop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(thiophen-3-yl)acetamide
N-[(3-methyloxetan-3-yl)methyl]-3-[(1,3-thiazol-2-ylmethyl)sulfamoyl]benzamide
methyl (2S,4S)-4-(4-methylbenzamido)-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidine-2-carboxylate
N-(3-cyanophenyl)-4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidine-1-carboxamide
1-(1-ethyl-1H-pyrazole-4-carbonyl)-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-{[3-(2-chlorophenyl)pyrrolidin-1-yl]methyl}-1-ethyl-3,5-dimethyl-1H-pyrazole
4-[(2-fluorophenyl)methyl]-1-[(trimethyl-1H-pyrazol-4-yl)methyl]piperidine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepane
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(6-methylpyridin-2-yl)methyl]amine
4-[3-(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidin-1-yl]-4-oxo-N-(1,3,4-thiadiazol-2-yl)butanamide
1-(oxan-4-ylmethyl)-6-(pyridin-2-ylmethoxy)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
2-[4-(2-methoxyethyl)piperazin-1-yl]-2-(6-methoxynaphthalen-2-yl)acetic acid
9-(4-ethylbenzoyl)-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-[(2-aminopyridin-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxylic acid
3-cyclohexyl-N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1H-pyrazole-4-carboxamide
dimethyl({4-methyl-5-[1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl]-4H-1,2,4-triazol-3-yl}methyl)amine
2,3-dimethyl-N,N-bis(1,3-oxazol-4-ylmethyl)quinoxaline-6-carboxamide
3-[(3R,4S)-3-(5-chlorofuran-2-amido)-4-propylpyrrolidin-1-yl]propanoic acid
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-propylacetamide
1-{3-[(3,4-dimethoxyphenyl)amino]piperidin-1-yl}-3-methoxypropan-1-one
5-cyclobutyl-N-[(6-methylquinolin-5-yl)methyl]-1,3,4-oxadiazol-2-amine
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-methyl-N-(1,2-oxazol-3-ylmethyl)propanamide
(3aS,6aR)-5-[(2,3-difluorophenyl)methyl]-3-[2-(4-methoxyphenyl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-(4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-3-methyl-1H-pyrazol-1-yl)ethan-1-ol
3-(1,2-oxazinan-2-yl)-N-[(1R,4S,6S)-spiro[bicyclo[2.2.1]heptane-7,1'-cyclopropan]-2-en-6-ylmethyl]propanamide
2-(2-chlorophenoxy)-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
5-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]sulfonyl}-2,3-dihydro-1,3-benzoxazol-2-one
4-(3-chlorophenoxy)-1-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperidine
5-(5-methylfuran-2-yl)-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1,2,4-triazin-3-amine
9-{[4-(2-aminoethyl)phenyl]methyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-methyl-2-{6-[(piperidin-4-yl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}phenol
3-(3-fluorophenyl)-N-methyl-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}benzamide
N-(1,2-oxazol-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-amino-3-ethyl-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(thiophen-3-yl)acetamide
methyl 5-({2-methyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-carboxylate
(3S,5S,9R)-5-{[(4-tert-butylphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
5-(2H-1,3-benzodioxol-5-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[3-(propan-2-yloxy)propyl]acetamide
2-(1-{[(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
4-{6-[(2-methoxyethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine