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N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-2-[3-(2-fluorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
N-[(3S)-2-oxoazepan-3-yl]-4-(2-oxopyrrolidin-1-yl)-N-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}benzamide
2-chloro-N-ethyl-4-({[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]carbamoyl}amino)benzamide
methyl 3-(4-chlorobenzoyl)-9-[3-(1-methyl-1H-pyrazol-4-yl)propoxy]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-(3-methyl-5-oxo-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-4-yl)-N-[3-(pyridin-3-yloxy)propyl]acetamide
3-(5-methylthiophen-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
3-fluoro-N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)benzamide
2-(morpholin-3-yl)-N-(4-{[2-(pyridin-2-yl)ethyl]sulfanyl}phenyl)acetamide
1-{3-[2-(2-fluorophenyl)ethyl]piperidin-1-yl}-2-methoxyethan-1-one
4-{4-[2-(3-fluorophenyl)acetamido]-1H-pyrazol-1-yl}-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
methyl 3-(2-methoxyacetamido)-1-methyl-5-(propylamino)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[2-(2-methoxyphenyl)ethyl]-6-{[4-(pyrrolidin-1-yl)phenyl]methyl}-6-azaspiro[2.5]octane-1-carboxamide
4-(1-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperidin-4-yl)pyridine
3-(2,4-dimethoxybenzoyl)-1-[(2-methylphenyl)methyl]piperidine
3-(azepane-1-carbonyl)-N-[(3-methoxyphenyl)methyl]-N-methyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(2,6-dimethylpyridin-3-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrimidin-2-amine
3-[2-(dimethylamino)ethyl]-8-[(2-methoxyquinolin-3-yl)methyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(2-ethoxyethyl)-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
(2R,6S)-4-[6-(3-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-2,6-dimethylmorpholine
N-[2-({[3-(hydroxymethyl)-2,4,6-trimethylphenyl]methyl}amino)ethyl]pyridine-4-carboxamide
5-{2-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-oxoethyl}-3,4-dihydropyrimidin-4-one
6-{4-[(1R,5S)-6-azabicyclo[3.2.1]octan-6-yl]piperidin-1-yl}pyridine-3-carbonitrile
(4aS,8aR)-6-[(2-methyl-1,3-oxazol-4-yl)methyl]-1-(piperidin-4-ylmethyl)-decahydro-1,6-naphthyridin-2-one
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-(dimethylamino)propanamide
(3R,4S)-1-[(2,6-dichloro-3-hydroxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(2-methylphenyl)propan-1-one
ethyl 1-(cyclohex-1-ene-1-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-2-(2-oxo-4-phenylpyrrolidin-1-yl)-N-(pyridin-4-ylmethyl)acetamide
(1R,5S)-6-methyl-3-[2-(pyridin-2-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
5-fluoro-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]quinazolin-4-amine
1-methyl-3-(thiomorpholine-4-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-methoxy-6-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)phenol
(butan-2-yl)({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(pyridin-4-ylmethyl)amine
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N,N-bis(pyridin-3-ylmethyl)acetamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}benzamide
6-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N-ethylpyridine-3-carboxamide
5-cyclopropyl-N-[2-(morpholin-4-yl)ethyl]-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carboxamide
ethyl 4-benzyl-1-(quinolin-5-ylmethyl)piperidine-4-carboxylate
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-[4-ethoxy-3-(hydroxymethyl)phenyl]pyridine-3-carbonitrile
4-chloro-1-ethyl-N-{2-[(pyridin-3-yl)amino]ethyl}-1H-pyrazole-3-carboxamide
6-[2-(3-methylpiperidin-1-yl)ethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
9-[(2,5-difluorophenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-cyclohexyl-5-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,2-oxazole-3-carboxamide
5-(4-chlorophenyl)-N-[2-(3-fluorophenyl)ethyl]-1,2,4-triazin-3-amine
2-fluoro-6-{4-[4-(propan-2-yl)piperazin-1-yl]phenyl}benzamide
ethyl 4-{1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-5-methyl-1H-pyrazole-4-amido}piperidine-1-carboxylate
ethyl 3-benzylpiperidine-3-carboxylate
(1S,5R)-3-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(4-fluorophenoxymethyl)-N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-1,3-oxazole-4-carboxamide