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(1R,3S)-3-methoxy-7-(2-methyl-1,3-benzothiazole-5-carbonyl)-7-azaspiro[3.5]nonan-1-ol
(3-benzyl-1H-1,2,4-triazol-5-yl)(4-methoxyphenyl)methanol
methyl (1R,3S,3aR,6aS)-5-ethyl-4,6-dioxo-3-[3-(trifluoromethyl)phenyl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
[(3R,5R)-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(2,1,3-benzothiadiazol-5-ylmethyl)({[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl})methylamine
4-[(2-methylprop-2-en-1-yl)oxy]-N-[(5-oxopyrrolidin-2-yl)methyl]-N-(propan-2-yl)benzamide
1-[7-(2,6-dimethoxyphenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
7-chloro-1-methyl-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1H-indole
1-{[5-(2-methylpropyl)-1H-pyrazol-3-yl]methyl}-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]acetamide
N-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 3-(1,3-dimethyl-1H-pyrazole-5-amido)-5-{[2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)acetamido]methyl}benzoate
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-3-ylmethyl)amino]methyl}piperidin-2-one
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-2-[(2-methoxyethyl)(methyl)amino]ethan-1-one
2-[5-(methoxymethyl)-3-[(2-methoxyphenyl)methyl]-1H-1,2,4-triazol-1-yl]ethan-1-ol
3-(1-{[3-(2,5-dimethylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-N-(2-methoxyethyl)propanamide
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(4,5,6,7-tetrahydro-2H-indazol-3-yl)propanamide
1-[2-(dimethylamino)ethyl]-3-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-3-(2-methylphenyl)pyrrolidine-2,5-dione
9-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3-oxa-9-azaspiro[5.5]undecane
(2S,4S)-4-amino-1-methyl-N-{3-oxo-3-[4-(propan-2-yl)piperazin-1-yl]propyl}pyrrolidine-2-carboxamide
N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}[2-(3-fluorophenyl)ethyl]amine
N-[(3R,5S)-1-(cyclohexylmethyl)-5-(diethylcarbamoyl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
5-(2-methoxyethyl)-3-(4-phenylphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
1-(3-methoxypropyl)-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-(2,5-dimethoxyphenyl)-N-{[7-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-methyl-2-[1-methyl-2,5-dioxo-3-(4-phenylphenyl)pyrrolidin-3-yl]-N-[(3-methylpyridin-2-yl)methyl]acetamide
6-ethyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-oxo-1,2-dihydropyridine-4-carboxamide
1-(1-benzylpyrrolidin-3-yl)-3-(1-methyl-1H-1,2,3-triazol-4-yl)urea
N-(3-ethyl-4-methyl-1-phenyl-1H-pyrazol-5-yl)-2-(1H-1,2,3-triazol-1-yl)acetamide
N-methyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]quinoline-8-carboxamide
4-[(3-fluorophenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-butyl-8-(2-ethylbutanoyl)-1,3,8-triazaspiro[4.5]dec-1-en-4-one
4-{[1-(cyclohexylmethyl)-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}morpholine
5-{1-[3-(2-methoxyphenyl)propanoyl]piperidin-4-yl}-5-propyl-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-methyl-N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(1H-imidazol-1-ylmethyl)piperidin-4-ol
4-(dimethyl-1,3-oxazole-5-carbonyl)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-{2-[(2,6-dimethylphenyl)carbamoyl]phenyl}oxane-4-carboxamide
4-cyano-N-(3-methoxypropyl)-1-methyl-N-[(4-methylphenyl)methyl]-1H-pyrrole-2-carboxamide
2-({[2-(dimethylamino)ethyl](thiophen-3-ylmethyl)amino}methyl)-6-methylphenol
(1S,5R)-3-methyl-6-(5-methyl-1,2-oxazole-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)amino]methyl}-2,6-dimethylphenol
2-acetamido-N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-3-hydroxypropanamide
3-[(4aR,7aS)-4-[2-(3-methylphenyl)acetyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]ethyl}urea
2-(4-fluorophenyl)-4-(5-phenyl-1,3-oxazole-4-carbonyl)morpholine
N-[(3S,4R)-1-{[4-methoxy-3-(methoxymethyl)phenyl]methyl}-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]acetamide