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1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)-1,4-diazepan-5-one
N-{5-[2-(3-methylphenoxy)ethyl]-1,3,4-thiadiazol-2-yl}-2-(1H-pyrazol-1-yl)butanamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
methyl 2-[benzyl(methyl)sulfamoyl]-6-(3-methylbutyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{1-[5-(4-fluorophenyl)-1,2,4-triazin-3-yl]piperidin-4-yl}-2-methylpropan-1-ol
2-{5H,6H,7H-cyclopenta[b]pyridin-3-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
N-[(2,3-dimethoxyphenyl)methyl]-5-(2,6-dimethylphenoxymethyl)-1,2-oxazole-3-carboxamide
2-{3-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidine-1-carbonyl]phenoxy}acetamide
{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}(methyl)(2-phenoxyethyl)amine
4-methyl-N-[2-(3-phenylpiperidin-1-yl)ethyl]-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
5-[3-(1H-imidazol-1-ylmethyl)piperidine-1-carbonyl]-N-(oxan-4-yl)pyridin-2-amine
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-methoxy-N-(1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
(1R,5R)-6-methyl-3-[2-(prop-2-en-1-yloxy)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
3-(2-oxopyrrolidin-1-yl)-N-{[5-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}benzamide
N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-5-[(methylsulfanyl)methyl]furan-2-carboxamide
2-[(5-ethyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-[1-(4-fluorophenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-(3-{[2-(4-chlorophenyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
4-(1-ethyl-1H-imidazol-2-yl)-1-(3-phenoxybenzoyl)piperidine
4-{[3-(benzyloxy)phenyl]methyl}-9-methoxy-7-(6-methoxypyridazin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-5,5-diphenylpiperidin-2-one
N-{[7-(4-cyclopropanecarbonylphenyl)-4-fluoro-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(thiophen-2-yl)acetamide
1-{2-[2-(6-chloro-2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-4-methyl-1H-1,2,3-triazole
1-[(3R)-3-hydroxypyrrolidin-1-yl]-2-(2,3,6-trimethylphenoxy)ethan-1-one
1-(4-methyl-1H-pyrrole-2-carbonyl)-4-[(3-methylpyridin-2-yl)methyl]piperazine
3-(2,3-dihydro-1-benzofuran-7-yl)-5-[(propan-2-yl)sulfamoyl]benzoic acid
N-[3-(4,6-dimethoxypyrimidin-2-yl)phenyl]acetamide
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-5-methyl-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-{methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}-N-(thiophen-2-ylmethyl)propanamide
3-(2,3-dihydro-1H-inden-2-yl)-5-(1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-4-yl)-5-methylimidazolidine-2,4-dione
3-methoxy-N-(2-methoxyethyl)-N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)propanamide
N-methyl-3-{methyl[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-(dimethylamino)pyridine-3-carboxamide
1-(azocan-1-yl)-3-[2-methoxy-4-({[2-(pyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
(3aR,7aS)-2-(pyridine-4-carbonyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
4-(2-methoxyethyl)-1-{[3-(2-methylphenyl)phenyl]methyl}-1,4-diazepan-5-one
2-(dimethylamino)-2-(4-fluorophenyl)-N-[2-(trimethyl-1H-pyrazol-1-yl)ethyl]acetamide
1-(3-methoxyphenyl)-6-methyl-4-(3-methylbutyl)piperazin-2-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-2-(2,3,6-trifluorophenyl)acetamide
6-[(3,5-dimethoxyphenyl)methoxy]-4-[(4-hydroxyphenyl)methyl]-1-(propan-2-yl)-1,4-diazepan-2-one
1-{[3-(1-benzofuran-2-yl)-1H-pyrazol-4-yl]methyl}-4-(thiophene-2-carbonyl)piperazine
1-[1-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]cyclopentanamine
4-[2-(dimethylamino)-2-(3-methylphenyl)acetyl]-N,N-dimethylpiperazine-1-carboxamide
1-{4-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]phenyl}-1H-imidazole
(1S,5R)-6-(cyclobutylmethyl)-3-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane