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1-(2,3-dihydro-1H-inden-2-yl)-4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-1,4-diazepane
N-(2-methoxyethyl)-2-(4-oxo-3,4-dihydroquinazolin-3-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
2-[2-(ethylsulfanyl)ethyl]-5-(piperidin-1-yl)-2,3-dihydropyridazin-3-one
1-{furo[3,2-c]pyridin-4-yl}-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
4-{[5-methyl-5-(4-methylpent-3-en-1-yl)-2-oxopiperidin-1-yl]methyl}benzene-1-sulfonamide
4-{[3-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-2-methyl-1,3-benzothiazole-5-carboxamide
5-(4-chlorophenyl)-3-[4-(2-methoxyphenoxy)piperidin-1-yl]-1,2,4-triazine
N-[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-amine
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-2-[(2-methylprop-2-en-1-yl)oxy]benzamide
3-(4-chlorobenzoyl)-1-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidine
(1S,5R)-6-benzyl-3-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-chloro-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}thiophene-2-carboxamide
4-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-N-methylpyridin-2-amine
1'-[2-(4-methyl-1,4-diazepan-1-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-({[1-({6-chloroimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidin-3-yl]oxy}methyl)pyridine
4-hydroxy-2-methyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}pyrimidine-5-carboxamide
N-(pyrrolidin-3-yl)-3-[(thiophen-3-ylmethyl)sulfamoyl]benzamide
N-(3,5-dimethoxyphenyl)-3-{1-[2-(1H-pyrazol-1-yl)acetyl]piperidin-3-yl}propanamide
4-(6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1-phenylpiperazin-2-one
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-N-[2-(pyridin-3-ylformamido)ethyl]acetamide
2-methoxy-6-[2-(pyridin-2-yl)-1H-imidazol-1-yl]pyridine
1-[(4-methoxy-2-methylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-{4-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}butanamide
5-[3-(4-fluorophenyl)-1H-pyrazol-5-yl]-3-[(methylsulfanyl)methyl]-1,2,4-oxadiazole
2-(4-methoxyphenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
1-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-4-(pyrrolidine-1-sulfonyl)piperazine
1-[2-(morpholine-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]isoquinoline
{3-[2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]propyl}dimethylamine
N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-3-(3-hydroxy-3-methylbutyl)benzamide
1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}-4-(pyrrolidine-1-sulfonyl)-1,4-diazepane
ethyl 1-[(3-{[1-(2-cyclopentylacetyl)piperidin-4-yl]oxy}phenyl)methyl]piperidine-2-carboxylate
5-methyl-5-(4-methylpent-3-en-1-yl)-1-[3-(1H-1,2,3-triazol-1-yl)propyl]piperidin-2-one
6-methyl-N-[(2-phenoxypyridin-3-yl)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-benzyl-8-(1-hydroxypropan-2-yl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[1'-(1-ethyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]-2-methoxyethan-1-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
1-[(1-cyclopentyl-5-oxopyrrolidin-3-yl)methyl]-3-(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
4'-(2,2-dimethylpropyl)-1-(furan-2-ylmethyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
6-[1-(cyclohexylmethyl)-3-methyl-1H-1,2,4-triazol-5-yl]-1,2,3,4-tetrahydroquinoxaline-2,3-dione
N-(2-methylpropyl)-1-(4,6,7-trimethylquinazolin-2-yl)piperidine-4-carboxamide
1-{3-[4-(2-methoxyphenyl)-3-oxopiperazin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]propanamide
6-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-3,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
N4,5-dimethyl-N4-[3-(pyrrolidin-1-yl)butyl]pyrimidine-2,4-diamine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-N-methyl-6-phenylimidazo[2,1-b][1,3]thiazole-3-carboxamide
1-[4-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(oxan-2-ylmethoxy)ethan-1-one
1-(2-butyl-1,3-benzoxazole-5-carbonyl)piperidin-4-ol
4-cyclobutyl-6-methyl-N-[1-(4-methylpyridin-2-yl)propyl]pyrimidin-2-amine
6-{3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carbonitrile