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N-[3-(2-methyl-1H-imidazol-1-yl)propyl]-2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-[4-(3-methoxybenzoyl)piperazin-1-yl]-5-phenyl-1,2,4-triazine
N-(3-cyano-4-ethoxyphenyl)-4-[2-(morpholin-4-yl)ethyl]piperazine-1-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]pyrazolo[1,5-a]pyridine-2-carboxamide
4-[(dimethylamino)methyl]-1-(2,3,6-trimethylquinoline-4-carbonyl)azepan-4-ol
[(3R,4S)-4-[(4-methylpiperazin-1-yl)methyl]-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]methanol
N-ethyl-3-propyl-N-(pyridin-4-ylmethyl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-N3-ethyl-N3-(2-methylprop-2-en-1-yl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
5-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyrazin-2-ol
{1-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
(3S)-1-[2-(2-phenylethyl)-1,3-benzoxazole-5-carbonyl]pyrrolidin-3-ol
N-ethyl-2-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}piperazin-1-yl)acetamide
2-[5-(6-methyl-2-phenylpyrimidin-4-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
(1-{[5-(1-benzofuran-5-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}piperidin-4-yl)methanol
3-[3-(propan-2-yloxy)benzoyl]-1-(thian-4-yl)piperidine
N-(1-{1-[(5-ethylfuran-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
{3-[4-(3-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-5-methyl-1,2-oxazol-4-yl}methanol
2-[3-(propan-2-yl)-5-{1-[2-(propan-2-yl)-1H-imidazol-1-yl]ethyl}-1H-1,2,4-triazol-1-yl]pyridine
N-[(2-chlorophenyl)methyl]-3-[1-(5-methylpyrazine-2-carbonyl)piperidin-3-yl]propanamide
2-(7-fluoro-2-methyl-1H-indol-3-yl)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}acetamide
(2S,4R)-N-[2-(2-chlorophenyl)ethyl]-4-(4-cyanobenzamido)pyrrolidine-2-carboxamide
4-[1-(2,5-dimethoxybenzoyl)piperidin-4-yl]pyridine
2-(1-cyclopentyl-4-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperazin-2-yl)ethan-1-ol
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-4-(4H-1,2,4-triazol-4-yl)benzamide
phenyl (7S,9aR)-7-(1H-indol-3-ylmethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
dimethyl({[3-methyl-7-(thiophene-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}sulfamoyl)amine
methyl 2-{[(1-methylpiperidin-3-yl)methyl](2-phenylethyl)carbamoyl}benzoate
2-[3-(2-chlorophenyl)-1-(2-methoxyethyl)-2,5-dioxopyrrolidin-3-yl]-N-ethyl-N-(2-methylprop-2-en-1-yl)acetamide
1-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-phenylethane-1,2-dione
4-({5-[1-(3-methoxypropyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
1-[4-(2-cyclobutyl-5-fluoro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-2-ethylbutan-1-one
4-methyl-2-(propan-2-yl)-5-(3-propoxypiperidine-1-carbonyl)pyrimidine
3-[2-({1-[3-(furan-2-yl)phenyl]piperidin-4-yl}amino)ethyl]-1,3-oxazolidin-2-one
1-(3-aminoazepan-1-yl)-3-(4-chloro-1H-pyrazol-1-yl)propan-1-one
3-[(3S,4R)-1-[(2-chlorophenyl)methyl]-4-[4-(2-fluorophenyl)piperazin-1-yl]piperidin-3-yl]-N-(2,4-dimethoxyphenyl)propanamide
3-(1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-[2-(dimethylamino)ethyl]-9-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
5-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazine-1-carbonyl}-1-[2-(pyridin-2-yl)ethyl]piperidin-2-one
1-[3-(methylsulfamoyl)phenyl]-3-(2,2,2-trifluoroethyl)urea
N-({1-[(2,3-difluoro-4-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-hydroxyacetamide
4-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-2-[1-(2-methoxyethyl)-1H-1,2,3,4-tetrazol-5-yl]morpholine
(3S,4R)-3-benzyl-1-(4-hydroxy-3-methoxybenzoyl)-4-methylpiperidin-4-ol
N-[2-(dimethylamino)ethyl]-5-(quinoxalin-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(5S,9aS,9bS)-5-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-2-(pyridin-3-ylmethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-[1-(3-fluorobenzoyl)piperidin-4-yl]-3-phenylpropan-1-ol
(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(1,3-thiazole-4-carbonyl)pyrrolidine-2-carboxamide
2-methoxy-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]quinoline-4-carboxamide
2-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]pyridine-3-carboxamide
N-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-2,3-difluoro-4-methoxybenzamide