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N-[(5-methylthiophen-2-yl)methyl]-N-(pyridin-2-ylmethyl)morpholine-2-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-2-(pyridin-3-yl)acetamide
11-{[(4-methylphenyl)methyl]amino}-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
6-fluoro-2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}quinolin-4-ol
3-methyl-7-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-{1-[1-(2-propoxyethyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-[(2-methylpyridin-3-yl)oxy]-1-(pyrimidin-2-yl)piperidine-4-carboxylic acid
N-(1H-1,3-benzodiazol-2-ylmethyl)-6-(2,5-dimethoxyphenyl)-N-methyl-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridine-3-carboxamide
N-(1-{7-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}-2-methylpropyl)-4-methoxybenzamide
1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-cyclohexyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
(1S,5R)-6-(5-chlorothiophene-2-carbonyl)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[5-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1,3-thiazol-2-yl]morpholine
2-{spiro[2.5]octan-1-yl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
methyl 2-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidine-1-carbonyl}benzoate
1-(4-hydroxyphenyl)-N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-5-oxopyrrolidine-3-carboxamide
(2S,4S)-N-ethyl-1-(1H-indol-5-ylmethyl)-4-[2-(methylsulfanyl)acetamido]pyrrolidine-2-carboxamide
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[(3-methylpyridin-2-yl)methyl]-N-(propan-2-yl)acetamide
4-fluoro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-methyl-N-(pyridin-4-ylmethyl)benzamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-2,3-dimethylquinoxaline-6-carboxamide
N-cyclobutyl-2-(2-hydroxypropanoyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-[(4-chlorophenyl)methyl]-N-(1-hydroxy-2-methylpropan-2-yl)-6-oxopiperidine-3-carboxamide
2-{2-[2-(furan-2-yl)azepan-1-yl]-2-oxoethyl}-2,3-dihydro-1,2-benzothiazol-3-one
2-[2-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
1-(oxane-4-carbonyl)-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-[5-(2,6-dimethylphenyl)-4-phenyl-1H-imidazol-1-yl]-1-(pyrrolidin-1-yl)propan-1-one
1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]-2-[(2-ethyl-6-methylpyridin-3-yl)oxy]ethan-1-one
3-(3-fluorophenyl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]-1H-pyrazole-4-carboxamide
1-[4-({[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}amino)piperidin-1-yl]ethan-1-one
2-benzyl-8-[2-(2-methoxyethoxy)acetyl]-2,8-diazaspiro[4.5]decan-3-one
{1-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
5-(methoxymethyl)-N-{[4-(3-methoxyphenyl)-5-[(2-phenylethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}furan-2-carboxamide
3-[1-(3,5-dimethyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-N-(5-hydroxypentyl)-2-(4-methylphenyl)acetamide
1-methyl-4-{5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-yl}piperazine
6-(2-chlorophenyl)-N-(oxan-4-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
3-{2-[4-(4-acetylphenyl)piperazin-1-yl]-2-oxoethyl}-3-(2-fluorophenyl)-1-(2-methoxyethyl)pyrrolidine-2,5-dione
(1S,3R)-3-amino-N-(5-chloro-2-ethyl-3-methyl-1-benzofuran-7-yl)cyclopentane-1-carboxamide
3-{2-[1-(3-aminothiophene-2-carbonyl)piperidin-2-yl]ethyl}phenol
4-methyl-1-(3-{3-oxo-3-[4-(pyridin-2-yl)piperazin-1-yl]propyl}piperidin-1-yl)pentan-1-one
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
4-(4-fluorophenoxy)-1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](ethyl)[2-(1H-pyrazol-1-yl)ethyl]amine
11-({[2-fluoro-4-(trifluoromethyl)phenyl]methyl}amino)-4-(pyridin-2-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)thiophen-2-yl]ethan-1-one
1-{[2-methanesulfonyl-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl}-4-phenyl-1,4-diazepane
4-[4-(piperidine-1-carbonyl)piperidin-1-yl]-2-[(trimethyl-1H-pyrazol-4-yl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione