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N-(1-benzylpiperidin-3-yl)-2-{[6-(pyrrolidin-1-yl)pyridazin-3-yl]oxy}acetamide
5-methyl-3-[3-(pyridin-2-ylmethyl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-2H-indazole
[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)(naphthalen-1-ylmethyl)amine
N-{[7-chloro-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-cyclopropylpropanamide
5-[2-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-2-oxoethyl]-1,3-dimethylimidazolidine-2,4-dione
2-{methyl[5-({methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}methyl)pyrimidin-2-yl]amino}acetic acid
5-(furan-2-yl)-1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-[2-(trifluoromethoxy)phenyl]pyridine-4-carbonitrile
2-(cyclopropylmethyl)-8-({4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-2,8-diazaspiro[5.5]undecan-3-one
4-benzyl-3-ethyl-N,N-dimethyl-5-oxo-1,4-diazepane-1-sulfonamide
N-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
2-(1-ethylpiperidin-4-yl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]acetamide
N-cyclopentyl-N'-(pyridin-2-ylmethyl)butanediamide
N-(1-cycloheptylpiperidin-3-yl)-2-(1-methylpiperidin-4-yl)acetamide
[4-(1H-1,2,3-triazole-5-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
5-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-5-[(2-fluorophenyl)methyl]imidazolidine-2,4-dione
N-[1-(4-tert-butylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-hydroxy-2-methylpropanamide
2-(2-oxobutyl)-5-(piperazin-1-yl)-2,3-dihydropyridazin-3-one
N-benzyl-N-methyl-3-({[3-(1H-pyrazol-1-yl)propyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-(4-chlorobenzoyl)-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine
4-(naphthalen-2-yl)-1-[2-(propan-2-yloxy)ethyl]-1H-1,2,3-triazole
{5-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methanol
5-phenyl-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-1,2,4-triazin-3-amine
2-[(4-{1-azabicyclo[2.2.2]octan-3-yl}piperazin-1-yl)methyl]benzoic acid
2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]-1,3-benzothiazole
4-{1H-pyrazolo[3,4-b]pyridin-4-yl}-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-({3,5-dimethoxy-4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)thiophene-2-carboxamide
methyl 4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrrole-2-carboxylate
7-(2,6-dimethoxyphenyl)-9-methoxy-4-[(4-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3-(pyridin-2-yl)propanamide
N-({3-[3-(trifluoromethyl)phenyl]-1,2,4-oxadiazol-5-yl}methyl)acetamide
3-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidine-1-carbonyl]phenyl}-1H-1,2,4-triazole
4-{[1-(dimethylsulfamoyl)piperidin-4-yl]oxy}-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
7-[(3,4-difluorophenyl)methyl]-2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-2,7-diazaspiro[4.5]decane
6-ethyl-2-methyl-4-[4-(pyridin-4-yl)piperidine-1-carbonyl]quinoline
2-{[cycloheptyl(pyridin-3-ylmethyl)amino]methyl}benzonitrile
1-cyclopentyl-4-(3-fluoropyridin-4-yl)-1,4-diazepane
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
[(3R,5R)-1-(5-methylthiophene-3-carbonyl)-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
(3aR,6aR)-2-methanesulfonyl-5-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
methyl 3-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-7-oxo-9-(3-phenylpropoxy)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(4-methoxynaphthalen-1-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[3-({[(3-methoxyphenyl)methyl]amino}methyl)-5-(piperidine-1-carbonyl)phenyl]methanesulfonamide
5-{1-[5-(2-chlorophenyl)furan-2-carbonyl]pyrrolidin-2-yl}-3-methyl-1,2-oxazole
N-(3-methyl-1-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)piperidine-4-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(2-methyl-1H-indol-1-yl)propanamide
1-(2,3-dihydro-1H-inden-5-yl)-5-[(2-methoxyethoxy)methyl]-3-(oxan-4-yl)-1H-1,2,4-triazole
2-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-1-[4-(benzyloxy)piperidin-1-yl]ethan-1-one