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3-(azepane-1-carbonyl)-N-ethyl-N-(2-methylprop-2-en-1-yl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-{[1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperidin-3-yl]methyl}thiophene-2-sulfonamide
N-[2-(1-hydroxycyclopentyl)ethyl]-N-methyl-1H-1,2,4-triazole-5-carboxamide
1-{1-[(3-methoxyphenyl)methyl]piperidin-4-yl}-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide
2-[1-(cyclohexylmethyl)-4-[(1-ethyl-1H-imidazol-2-yl)methyl]piperazin-2-yl]ethan-1-ol
4-[3-(furan-2-yl)-1H-pyrazol-1-yl]-1-(5-methylthiophene-2-carbonyl)piperidine-4-carboxylic acid
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-ethyl-5-[1-(3-phenylpropyl)piperidin-4-yl]imidazolidine-2,4-dione
N-(5-{4-[(dimethylcarbamoyl)methyl]piperazine-1-carbonyl}-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-2,3-dimethylbenzamide
N-(2-{imidazo[1,2-a]pyridin-3-yl}ethyl)-5-methoxyfuran-2-carboxamide
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
3-{[(5-oxopyrrolidin-2-yl)methyl]sulfamoyl}-N-(pyridin-3-yl)benzamide
(2S,4S)-4-{[(2,6-difluorophenyl)methyl]amino}-N-methyl-1-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
2-methyl-N-{[7-(naphthalen-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}butanamide
2-{1-[(4-fluorophenyl)methyl]-4-(quinolin-5-ylmethyl)piperazin-2-yl}ethan-1-ol
N-{2-[1-(4-methoxyquinazolin-6-yl)-1H-imidazol-4-yl]ethyl}acetamide
N-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-2,3,6-trimethylquinoline-4-carboxamide
5-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
1-benzyl-5-(7-methoxy-2H-1,3-benzodioxol-5-yl)-3-methyl-1H,4H-pyrazolo[3,4-d]imidazole
N-(2-{[(3-chlorophenyl)methyl]sulfanyl}ethyl)-2,7-dioxo-1,3-diazepane-4-carboxamide
1,3-dimethyl-6-({4-oxo-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-1'-yl}carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-{thieno[3,2-d]pyrimidin-4-yl}-1,4-oxazepan-6-ol
N-[(3S,4R)-1-{3-fluoro-7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-methoxy-2-phenyl-N-{1-[1-(4,4,4-trifluorobutanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}acetamide
1-(2-cyclohexylethyl)-3-hydroxy-3-({[(3-hydroxyphenyl)methyl](methyl)amino}methyl)piperidin-2-one
2-[3-cyclopropyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]-1,1,1-trifluoropropan-2-ol
4-[({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)methyl]-1-ethylpyrrolidin-2-one
8-[(2-methylphenyl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{2-[3-(pentan-3-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pyrimidin-4-yl}piperidin-3-ol
3-acetamido-N-(2-fluorophenyl)-5-{[(2-phenylpropyl)amino]methyl}benzamide
3-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-1,6-dimethyl-1,2-dihydropyridin-2-one
3-propyl-N-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-1H-pyrazole-5-carboxamide
N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-(2H-1,3-benzodioxol-5-yl)propanamide
6-methoxy-N-[2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)ethyl]pyrimidin-4-amine
N-butyl-N-(furan-2-ylmethyl)-6-(2-hydroxyethyl)pyrazolo[1,5-a]pyrimidine-2-carboxamide
5-acetyl-N,2,4-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrrole-3-carboxamide
5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-oxazole-3-carboxamide
N-[1-(2,3-dihydro-1H-inden-2-yl)-5-oxopyrrolidin-3-yl]pyridine-3-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(methylsulfanyl)propanamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(pentan-3-yl)-1,2-oxazole-3-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[methyl(thiophen-2-ylmethyl)amino]pyridine-3-carboxamide
1-[3-(3-methoxyphenoxymethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
1-cyclohexyl-3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-4-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,4-diazepane
3-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]-1-[2-(phenylsulfanyl)ethyl]urea
2-(2-{[methyl(thian-4-yl)amino]methyl}phenoxy)acetic acid
2-(6-methoxypyridin-3-yl)-4-(trifluoromethyl)pyrimidine
2-(1-methyl-1H-imidazol-2-yl)-1-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
2-[(1-acetylpiperidin-4-yl)oxy]-N-(2-hydroxy-2-phenylethyl)-5-methoxy-N-methylbenzamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
5-[(4-methanesulfonylphenyl)methyl]-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid