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(3aR,6aR)-2-cyclopentyl-N-[3-(pyridin-4-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
7-(2-methoxyethyl)-2-[3-(4-methylphenyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
3-[(1-benzylpiperidin-4-yl)methyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
5-(4-methoxyphenyl)-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]furan-2-carboxamide
3-[4-(2-methoxyethoxy)piperidin-1-yl]-5-(5-methylfuran-2-yl)-1,2,4-triazine
3-{5-[2-(3-chloro-4-hydroxyphenyl)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-{[3-(2,5-dimethoxyphenyl)pyrrolidin-1-yl]methyl}-5-(1,5-dimethyl-1H-pyrrol-2-yl)-1,3,4-oxadiazole
methyl 2-[(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazol-3-yl)formamido]-4-(methylsulfanyl)butanoate
1-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
methyl 3-[(2E)-3-phenylprop-2-enamido]-5-[(pyridin-3-ylformamido)methyl]benzoate
1-(2-{[(4-{1-azabicyclo[3.2.1]octan-5-yloxy}phenyl)methyl]amino}ethyl)imidazolidin-2-one
[5-(1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methanol
4-(1-{[methyl(propan-2-yl)carbamoyl]methyl}piperidin-3-yl)benzoic acid
N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(3-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
(3R,4R)-1-[2-(4-chlorophenoxy)ethyl]-4-(2-methoxyethyl)-3-methylpiperidin-4-ol
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
2-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-N-(2-ethylphenyl)-2-oxoacetamide
N-(butan-2-yl)-3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
5-{4-[(4-chlorophenyl)methyl]piperazine-1-carbonyl}isoquinoline
N-{3-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]phenyl}acetamide
methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})(thiophen-3-ylmethyl)amine
5-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-6-methyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-methyl-N-propyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
6-chloro-N,N-dimethyl-3-({[2-phenyl-2-(piperidin-1-yl)ethyl]amino}methyl)imidazo[1,2-a]pyridine-2-carboxamide
[(2-{furo[3,2-c]pyridin-4-yloxy}phenyl)methyl]dimethylamine
N-ethyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
(3aR,6aR)-N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-methyl-4-{[(2-methylquinolin-5-yl)carbamoyl]amino}butanamide
6-(2H-1,3-benzodioxol-4-ylmethyl)-1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-6-azaspiro[2.5]octane
8-[(4-fluoro-2-methylphenyl)methyl]-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(4aS,7aR)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cycloheptyl-N-methyl-N-[(1-methylpyrrolidin-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-[(4-{[1-(furan-3-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]morpholine
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]ethan-1-one
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-1,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-(propan-2-yl)acetamide
ethyl 1-[5-fluoro-4-(morpholin-4-yl)pyrimidin-2-yl]piperidine-4-carboxylate
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(oxan-4-yl)acetamide
methyl 2-(4-{4-[(2-fluorophenyl)methyl]-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)benzoate
2-{[(3,3-diphenylpropyl)amino]methyl}-4-(pyrimidin-2-yl)phenol
N-(4-fluoro-2-methylphenyl)-3-[1-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)piperidin-3-yl]propanamide
6-(1-benzofuran-2-ylmethyl)-N-[2-(cyclohex-1-en-1-yl)ethyl]-6-azaspiro[2.5]octane-1-carboxamide
2-({3-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}methyl)-1H-1,3-benzodiazole
1-methyl-4-{2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]-2-oxoethyl}-2,3,4,5-tetrahydro-1H-1,4-benzodiazepine-2,5-dione
ethyl N-{[(2S,4S)-4-fluoro-1-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}pyrrolidin-2-yl]methyl}carbamate
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carbonyl}piperidine