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3-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-4-phenylpyridine
N-(3-methoxyphenyl)-3-[1-(3-phenyl-1,2-oxazole-5-carbonyl)piperidin-4-yl]propanamide
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-{5-[2-(2-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}-N-methylpropanamide
4-{1-[2-(2H-1,3-benzodioxol-5-yl)-1H-imidazol-1-yl]ethyl}-2-fluorophenol
2-({4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}methyl)-6,8-dimethylquinolin-4-ol
N-[(1-cyclooctylpyrrolidin-3-yl)methyl]-2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)acetamide
5-methoxy-2-{[3-(naphthalene-2-carbonyl)piperidin-1-yl]methyl}-4H-pyran-4-one
1-[6-(3-fluoro-4-methoxyphenyl)imidazo[2,1-b][1,3]thiazole-3-carbonyl]-1,4-diazepan-5-one
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-3-(trimethyl-1H-pyrazol-4-yl)propanamide
3-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]propanamide
4-[3-(trifluoromethoxy)phenyl]-1H-imidazole
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-methylpiperidine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-3-ethyl-1H-pyrazole-5-carboxamide
methyl 4-(4-{[4-(4-chlorophenoxy)piperidin-1-yl]methyl}-5-methyl-1,3-oxazol-2-yl)benzoate
4-{[3-(morpholine-4-carbonyl)-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}quinoline
N-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-4-(3-methylpyridin-4-yl)piperazine-1-carboxamide
(3aS,6aS)-2-[(2-aminopyridin-3-yl)methyl]-5-cyclobutanecarbonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
6-(dimethylamino)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylpyridine-3-carboxamide
(2R)-2-amino-N-[1-benzyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]propanamide
(1S,5R)-6-(dimethyl-1,3-oxazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
7-(2,6-difluoro-3-methylbenzoyl)-5H,6H,7H,8H-imidazo[1,5-a]pyrazine
N-[2-(3-methylpyridin-2-yl)ethyl]-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
methyl 6-[(4-hydroxyphenyl)methyl]-2-(1,2,3,4-tetrahydroisoquinoline-2-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[2-(1H-imidazol-4-yl)ethyl]-8-(2-methylpyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-N-(prop-2-en-1-yl)-3-(propan-2-yl)-1,2-oxazole-5-carboxamide
(1R,3S)-3-(2-aminoethoxy)-7-(2,3-dihydro-1H-inden-2-yl)-7-azaspiro[3.5]nonan-1-ol
2-({4-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)ethan-1-ol
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-2,5-dimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
7-methyl-6-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1H,2H-pyrazolo[1,5-a]pyrimidin-2-one
N-(2-phenylpropyl)-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
3,5-dimethyl-2-[1-(pyridin-3-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl]-1H-indole
5-[1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
1,3-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-N-propyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
1-{4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidine-1-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-3-(3-fluoro-4-phenylbenzoyl)piperidine-1-carboxamide
3-{1-oxaspiro[4.4]nonan-3-yl}-1-[4-(propylsulfamoyl)phenyl]urea
N-(2-methoxyethyl)-4-(1,3-thiazol-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-[4-(1H-imidazol-2-ylmethyl)piperazin-1-yl]-1,3-benzothiazole
2-(4-fluorophenyl)-4-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]morpholine
N-{3-[1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazol-5-yl]-2,5-dimethyl-1H-pyrrol-1-yl}acetamide
(2S,4S,5R)-1,2-dimethyl-5-(2-methylphenyl)-4-[(pyridin-4-ylmethyl)carbamoyl]pyrrolidine-2-carboxylic acid
(3aR,6aS)-5-methyl-N-[3-(2-methylpyrimidin-4-yl)phenyl]-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide
6-[3-(1H-1,2,4-triazol-1-yl)adamantan-1-yl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(5-methylfuran-2-yl)methyl]piperidine-4-carboxamide
1-ethyl-3-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]piperidine-3-carboxamide
N-(oxan-2-ylmethyl)-2-(4-phenylphenyl)acetamide
2-(4-acetylphenoxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}acetamide
(1S,4S)-2-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-2-azabicyclo[2.2.1]heptane
3-[2-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)ethyl]-1,3-oxazinan-2-one