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N-[(7R,8aS)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-dimethyl-1H-indole-5-carboxamide
1-(6-cyclopropylpyrimidin-4-yl)-3-[(2-fluorophenyl)methyl]piperidine-3-carboxylic acid
3-[methyl(2-{5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}pyrimidin-4-yl)amino]propane-1,2-diol
{4-benzyl-1-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
(3S,4R)-4-(hydroxymethyl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-ol
(1R,2R,6S,7S)-4-[3-(2-methyl-1H-imidazol-1-yl)propyl]-4-azatricyclo[5.2.1.02,6]decane
methyl 1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-4-carboxylate
1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
1-cyclopropyl-5-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]pyrrolidine-3-carboxamide
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
1-(1-{2-amino-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}piperidin-4-yl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-(1-{[4-(diethylamino)phenyl]methyl}piperidin-4-yl)-5-methyl-3-(thiophen-3-ylmethyl)imidazolidine-2,4-dione
2-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-4-methyl-1H-1,3-benzodiazole
N-(2-{3-[(6,7-dimethoxy-1,2,3,4-tetrahydroisoquinolin-2-yl)methyl]phenoxy}propyl)pyridine-2-carboxamide
1-(4-methylpiperidin-1-yl)-3-{[1-(1H-pyrazol-1-yl)propan-2-yl]amino}propan-1-one
3-[5-(phenoxymethyl)-3-(pyridin-3-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
3-(1H-1,3-benzodiazol-2-yl)-1-{3-[methyl(2-phenylethyl)amino]piperidin-1-yl}propan-1-one
N-[phenyl(pyridin-4-yl)methyl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]acetamide
N-(1-butyl-4-methyl-1H-pyrazol-5-yl)-2,3-dihydro-1,4-benzodioxine-2-carboxamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-(2-propoxyethyl)-1H-pyrazole-3-carboxamide
4,6-dimethyl-13-[(2E)-pent-2-en-2-yl]-3,7,8,10-tetraazatricyclo[7.4.0.02,7]trideca-1,3,5,8-tetraen-11-one
2-cyclohexyl-N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-1,3-benzoxazole-6-carboxamide
1-(4-ethylpiperazin-1-yl)-3-[4-({[(2-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
(3aR,6aR)-2-methanesulfonyl-5-{6,7,8,9-tetrahydro-5H-benzo[7]annulen-7-yl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[2-(methylsulfanyl)acetyl]-N-(oxolan-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
4-{[(4aS,7aR)-4-(2-carboxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]methyl}benzoic acid
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}furan-3-carboxamide
1-(1H-1,2,3-benzotriazol-5-yl)-3-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-methylurea
6,6-dimethyl-5-oxo-N-[2-(pyridin-2-ylsulfanyl)ethyl]thiomorpholine-3-carboxamide
3-(2-methoxyethyl)-5-(oxolan-3-ylmethyl)-1-(2-phenylethyl)-1H-1,2,4-triazole
(2R,3S,6R)-3-(2,3-difluorophenyl)-5-(4-methyl-1H-imidazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-cyclohexyl-N-[2-(1H-indol-3-yl)ethyl]-2-(morpholin-3-yl)acetamide
{2-[3-(2-hydroxyethyl)-4-[(3-methoxyphenyl)methyl]piperazin-1-yl]-2-oxoethyl}urea
N-cyclooctyl-2-[methyl({[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetamide
6-ethyl-N-[3-(1H-imidazol-1-yl)-1-phenylpropyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
2-methyl-4-[4-(2-methylpropyl)-3-oxo-6-(pyridin-3-ylmethoxy)-1,4-diazepane-1-carbonyl]-1,2-dihydrophthalazin-1-one
2,6-dimethoxy-4-({3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl}methyl)phenol
1-cyclopropyl-4-(3,3-diphenylpiperidine-1-carbonyl)pyrrolidin-2-one
2-(3-fluorophenyl)-6-(piperidin-4-yl)-3,4-dihydropyrimidin-4-one
N-{[7-(3-fluoro-4-methoxybenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-2-(methylsulfanyl)benzamide
1-(4-tert-butylbenzoyl)-N-ethyl-N-(pyridin-4-ylmethyl)piperidin-3-amine
1-[1-(1-ethyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
dimethyl(3-{2-[1-(pyridine-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}propyl)amine
1-[4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
2-(ethylsulfanyl)-1-[1-(hydroxymethyl)-9-(pyridin-4-ylmethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
3-(3-methoxyphenyl)-N-methyl-N-[2-(oxan-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2,6-dichloro-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
1-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-3-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}urea
(2S,4R)-4-(dimethylamino)-1-(5-ethylthiophene-3-carbonyl)pyrrolidine-2-carboxylic acid
1-(2,3-dihydro-1H-inden-2-yl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine